SCHEMBL988050

SCHEMBL988050

O=C(O)c1ccccc1-c1cc2cc(Cl)ccc2[nH]1

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.59
MEN1 O00255 2/20 0.59
NPC1 O15118 2/20 0.59
KMT2A Q03164 2/20 0.59
ALDH1A1 P00352 2/20 0.59
KDM4E B2RXH2 2/20 0.59
LMNA P02545 1/20 0.59
MAPT P10636 1/20 0.59
CYP19A1 P11511 1/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
NHERF1 O14745 1/20 0.56
F7 P08709 2/20 0.55
F3 P13726 2/20 0.55
FFAR1 O14842 10/20 0.50
PPARG P37231 2/20 0.50
GRIK1 P39086 1/20 0.44
DAO P14920 1/20 0.44
TP53 P04637 1/20 0.44
SIRT1 Q96EB6 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6439902 0.84 F2 (0.49) RAB9AALDH1A1KDM4ENHERF1F7
SCHEMBL27437769 0.83 KDR (0.56) RAB9AMEN1NPC1KMT2AALDH1A1
SCHEMBL25175575 0.80 KDM4E (0.62) RAB9AMEN1NPC1KMT2AALDH1A1
SCHEMBL28167722 0.79 MEN1 (0.61) RAB9AMEN1NPC1KMT2AALDH1A1
SCHEMBL11488198 0.79 MEN1 (0.61) RAB9AMEN1NPC1KMT2AALDH1A1
SCHEMBL17065800 0.77 MEN1 (0.63) RAB9AMEN1NPC1KMT2AALDH1A1
SCHEMBL26086683 0.76 F3 (0.50) RAB9AKDM4EF3DAO
SCHEMBL28763445 0.76 MEN1 (0.61) RAB9AMEN1NPC1KMT2AALDH1A1
SCHEMBL29808535 0.75 KDM4E (0.70) RAB9AMEN1NPC1KMT2AALDH1A1
SCHEMBL6117859 0.75 MEN1 (1.00) RAB9AMEN1NPC1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8598355-B2 Amide compound ASTELLAS PHARMA INC. (JP) 2013-12-03 US disclosed
EP-2565191-A1 4-(Indol-7-ylcarbonylaminomethyl)cyclohexanecarboxylic acid derivatives as EP4 receptor antagonists useful for the treatment of chronic renal failure or diabetic nephropathy Astellas Pharma Inc. (JP) 2013-03-06 EP disclosed
US-20110144153-A1 AMIDE COMPOUND ASTELLAS PHARMA INC. (JP) 2011-06-16 US disclosed
US-20110144153-A1 AMIDE COMPOUND ASTELLAS PHARMA INC. (JP) 2011-06-16 US disclosed
US-20110144153-A1 AMIDE COMPOUND ASTELLAS PHARMA INC. (JP) 2011-06-16 US disclosed
CN-102026961-A Amide compound ASTELLAS PHARMA INC 2011-04-20 CN disclosed
EP-2277858-A1 AMIDE COMPOUND Astellas Pharma Inc. (JP) 2011-01-26 EP disclosed
EP-2277858-A1 AMIDE COMPOUND Astellas Pharma Inc. (JP) 2011-01-26 EP disclosed
WO-2009139373-A1 AMIDE COMPOUND アステラス製薬株式会社 (JP) 2009-11-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110144153-A1 AMIDE COMPOUND PTGER4, PTGER1, PTGER2 RAB9A 3160/4885MEN1 4408/4885NPC1 2978/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.