SCHEMBL989277

SCHEMBL989277

CC1(C)CN=C(NCCCCCCCCCCCCNC2=NCCC2)NC1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 3/20 0.45
CYP2D6 P10635 1/20 0.38
TP53 P04637 1/20 0.37
RAB9A P51151 1/20 0.37
ALOX15 P16050 3/20 0.36
ALDH1A1 P00352 2/20 0.34
USP2 O75604 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.32
HSD17B10 Q99714 1/20 0.32
HTR1A P08908 1/20 0.31
HTR1D P28221 1/20 0.31
APOBEC3A P31941 1/20 0.31
APOBEC3G Q9HC16 1/20 0.31
POLB P06746 1/20 0.31
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL2418668 0.89 TP53 (0.40) CXCR4CYP2D6TP53RAB9AALOX15
SCHEMBL988394 0.86 CXCR4 (0.50) CXCR4APOBEC3AAPOBEC3G
Iodide SCHEMBL2419341 0.84 CXCR4 (0.49) CXCR4APOBEC3AAPOBEC3G
SCHEMBL988717 0.82 CXCR4 (0.44) CXCR4
SCHEMBL989088 0.76 CYP2D6 (0.53) CXCR4CYP2D6TP53RAB9AALOX15
Trifluoroacetic Acid SCHEMBL2419010 0.72 HRH4 (0.40) CXCR4
SCHEMBL12322123 0.64
SCHEMBL10925690 0.64
SCHEMBL10884472 0.64 CYP2D6 (0.71) CYP2D6TP53RAB9AALOX15ALDH1A1
Bromide SCHEMBL11659698 0.63 CYP2D6 (0.50) CYP2D6TP53RAB9AALOX15ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8012985-B2 parasiticides, in particularly against Plasmodium and babesia; antimalarial agents CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (C.N.R.S.) (FR) 2011-09-06 US disclosed
EP-2275100-A2 Compounds with anti-parasitic activity and drugs containing said compounds Centre National de la Recherche Scientifique (CNRS) (FR) 2011-01-19 EP disclosed
EP-2266555-A2 Compounds with antiparasitic activity and medicines containing same Centre National de la Recherche Scientifique (CNRS) (FR) 2010-12-29 EP disclosed
EP-2260840-A2 Compounds with antiparasitic activity and medicines containing same Centre National de la Recherche Scientifique (CNRS) (FR) 2010-12-15 EP disclosed
EP-2260841-A2 Compounds with antiparasitic activity and medicines containing same Centre National de la Recherche Scientifique (CNRS) (FR) 2010-12-15 EP disclosed