SCHEMBL9902003

SCHEMBL9902003

[NH]CCN1CCC(Oc2ccccc2C(F)(F)F)CC1

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SCD O00767 12/20 0.52
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
EPHX2 P34913 1/20 0.47
KDM4E B2RXH2 1/20 0.46
LMNA P02545 1/20 0.46
MAPT P10636 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
CARM1 Q86X55 1/20 0.46
PRMT6 Q96LA8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9902006 0.86 SCD (0.55) SCDCYP3A4CYP2D6
SCHEMBL5541389 0.86 SCD (0.52) SCDCYP3A4CYP2D6EPHX2KDM4E
SCHEMBL5541289 0.84 SCD (0.50) SCDCYP3A4CYP2D6EPHX2KDM4E
SCHEMBL5540517 0.83 SCD (0.54) SCDCYP3A4CYP2D6EPHX2
SCHEMBL5541771 0.83 SCD (0.49) SCDCYP3A4CYP2D6EPHX2KDM4E
SCHEMBL5543355 0.82 SCD (0.48) SCDCYP3A4CYP2D6EPHX2KDM4E
SCHEMBL5542451 0.81 KDM4E (0.64) SCDCYP3A4CYP2D6EPHX2KDM4E
SCHEMBL5542445 0.79 SCD (0.57) SCDCYP3A4CYP2D6EPHX2
SCHEMBL6819584 0.77 UTS2R (0.57) SCDCYP3A4CYP2D6KDM4ELMNA
SCHEMBL12099559 0.76 SCD (0.55) SCDCYP3A4CYP2D6EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2462121-A1 DERIVATIVES OF 2H PYRIDAZIN- 3 -ONES, THEIR PREPARATION AND THEIR USE AS SCD-1 INHIBITORS Pierre Fabre Médicament (FR) 2012-06-13 EP disclosed