SCHEMBL9902608

SCHEMBL9902608

O=c1cccnn1C(c1ccccn1)C(O)(c1cccnc1)c1cccnc1

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 14/20 0.45
KCNH2 Q12809 9/20 0.45
LMNA P02545 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
CYP19A1 P11511 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1243216 0.84 KCNA5 (0.50) KCNA5KCNH2
SCHEMBL1242038 0.83 KCNA5 (0.45) KCNA5KCNH2LMNACYP1A2CYP3A4
SCHEMBL1241829 0.83 KCNA5 (0.45) KCNA5KCNH2LMNACYP1A2CYP3A4
SCHEMBL1242003 0.83 KCNA5 (0.45) KCNA5KCNH2LMNACYP1A2CYP3A4
SCHEMBL9902593 0.81 KCNA5 (0.45) KCNA5KCNH2LMNACYP1A2CYP3A4
SCHEMBL1242831 0.81 KCNA5 (0.47) KCNA5KCNH2CYP19A1
SCHEMBL1242076 0.79 KCNA5 (0.48) KCNA5KCNH2CYP3A4CYP11B1CYP11B2
SCHEMBL1240403 0.75 KCNA5 (0.50) KCNA5KCNH2
SCHEMBL1242597 0.74 KCNA5 (0.40) KCNA5CYP1A2
SCHEMBL1242232 0.73 KCNA5 (0.50) KCNA5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781635-B1 POTASSIUM CHANNEL INHIBITORS MERCK SHARP & DOHME (US) 2012-06-13 EP disclosed