SCHEMBL9903689

SCHEMBL9903689

O=c1cc(O)ccn1C(c1ccc(F)cc1)C(O)(c1cccnc1)c1cccnc1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 11/20 0.45
KCNH2 Q12809 7/20 0.45
POLB P06746 1/20 0.37
CYP19A1 P11511 3/20 0.37
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
CYP3A4 P08684 2/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
CYP3A5 P20815 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1240347 0.86 KCNA5 (0.48) KCNA5KCNH2POLBCYP19A1CYP11B1
SCHEMBL1242868 0.85 KCNA5 (0.50) KCNA5KCNH2POLBCYP19A1CYP3A4
SCHEMBL9903505 0.81 KCNA5 (0.47) KCNA5KCNH2POLBCYP19A1CYP11B1
SCHEMBL9903168 0.80 KCNA5 (0.46) KCNA5KCNH2POLBCYP19A1CYP3A4
SCHEMBL1240425 0.78 KCNA5 (0.45) KCNA5KCNH2POLBCYP19A1CYP11B1
SCHEMBL1242076 0.77 KCNA5 (0.48) KCNA5KCNH2POLBCYP19A1CYP11B1
SCHEMBL1243603 0.77 KCNA5 (0.46) KCNA5KCNH2POLBCYP19A1CYP3A4
SCHEMBL1243497 0.77 KCNA5 (0.59) KCNA5KCNH2CYP3A4CYP2C9CYP2C19
SCHEMBL9902439 0.77 KCNA5 (0.59) KCNA5KCNH2CYP3A4CYP2C9CYP2C19
SCHEMBL1243006 0.76 KCNA5 (0.45) KCNA5KCNH2POLBCYP19A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781635-B1 POTASSIUM CHANNEL INHIBITORS MERCK SHARP & DOHME (US) 2012-06-13 EP disclosed