SCHEMBL9921365

SCHEMBL9921365

C[C@@H](Nc1ncnc2ccc([N+](=O)[O-])cc12)c1ccc(F)cc1

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EGFR P00533 10/20 0.59
DYRK1A Q13627 1/20 0.52
PIK3CA P42336 1/20 0.52
ALK Q9UM73 1/20 0.51
ALDH1A1 P00352 3/20 0.49
MAPT P10636 3/20 0.49
HTT P42858 3/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
GAA P10253 1/20 0.48
NCOA1 Q15788 1/20 0.48
NCOA3 Q9Y6Q9 1/20 0.48
CNR1 P21554 1/20 0.47
CNR2 P34972 1/20 0.47
GALR3 O60755 1/20 0.47
NR2F2 P24468 1/20 0.47
EIF2AK2 P19525 1/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9921351 1.00 EGFR (0.59) EGFRDYRK1APIK3CAALKALDH1A1
SCHEMBL28505293 0.93 EGFR (0.59) EGFRDYRK1APIK3CAALKALDH1A1
SCHEMBL13170964 0.90 GAA (0.57) EGFRALKALDH1A1MAPTHTT
SCHEMBL13170966 0.90 GAA (0.57) EGFRALKALDH1A1MAPTHTT
SCHEMBL7263353 0.88 EGFR (0.65) EGFRDYRK1APIK3CAALKALDH1A1
SCHEMBL13170962 0.88 EGFR (0.65) EGFRDYRK1APIK3CAALKALDH1A1
SCHEMBL7263343 0.88 EGFR (0.65) EGFRDYRK1APIK3CAALKALDH1A1
SCHEMBL28513093 0.85 HTT (0.59) EGFRALKALDH1A1MAPTHTT
SCHEMBL28509057 0.81 GALR3 (0.69) EGFRDYRK1AALDH1A1MAPTHTT
SCHEMBL24576686 0.80 EGFR (0.65) EGFRDYRK1APIK3CAHTTCNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012079079-A1 PRODUCTION OF INDUCED PLURIPOTENT STEM CELLS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2012-06-14 WO disclosed
WO-2011011522-A2 POTENT SMALL MOLECULE INHIBITORS OF AUTOPHAGY, AND METHODS OF USE THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2011-01-27 WO disclosed