SCHEMBL9921586

SCHEMBL9921586

Cc1cc(Cc2cnc(-c3nc4n(c(=O)c3O)CC3CCC4(NC(=O)c4ccn(C)n4)CC3)[nH]2)ccc1F

nearest known ligand 0.32

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14214203 0.96 GRIN1 (0.31) GRIN1GRIN2B
SCHEMBL9921559 0.89
SCHEMBL9905142 0.88 GRIN1 (0.31) GRIN1GRIN2B
SCHEMBL9921536 0.87 GRIN1 (0.34) GRIN1GRIN2B
SCHEMBL9921619 0.86
SCHEMBL9921571 0.85
SCHEMBL14214206 0.85
SCHEMBL14214200 0.83 GRIN1 (0.33) GRIN1GRIN2B
SCHEMBL14214199 0.82
SCHEMBL9921576 0.82 NTRK1 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8846659-B2 HIV integrase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2014-09-30 US disclosed
US-8846659-B2 HIV integrase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2014-09-30 US disclosed
WO-2012078844-A1 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-06-14 WO disclosed