SCHEMBL9923075

SCHEMBL9923075

Cc1ccccc1Nc1c(C(N)=O)cnn2c(N)ccc12

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 2/20 0.47
PDE4B Q07343 3/20 0.44
PDE4A P27815 2/20 0.41
PDE4C Q08493 2/20 0.41
PDE4D Q08499 2/20 0.41
SYK P43405 1/20 0.41
TYK2 P29597 2/20 0.41
CLCN2 P51788 1/20 0.40
TLR8 Q9NR97 1/20 0.39
NPC1 O15118 1/20 0.39
PKM P14618 1/20 0.39
RAB9A P51151 1/20 0.39
LMNA P02545 1/20 0.39
BRD4 O60885 1/20 0.39
BRD2 P25440 1/20 0.39
BRD3 Q15059 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9920270 0.89 CSF1R (0.48) CSF1RPDE4BPDE4APDE4CPDE4D
SCHEMBL9923079 0.85 CSF1R (0.45) CSF1RPDE4BPDE4APDE4CPDE4D
SCHEMBL12875308 0.83 CSF1R (0.44) CSF1RPDE4BPDE4APDE4CPDE4D
SCHEMBL1160648 0.83 PDE4B (0.48) CSF1RPDE4BPDE4APDE4CPDE4D
SCHEMBL9920282 0.80 JAK2 (0.58) TYK2NPC1RAB9A
SCHEMBL9920277 0.79 JAK3 (0.50) CSF1RTYK2
SCHEMBL9923398 0.74 JAK3 (0.47) CSF1RTYK2LMNA
SCHEMBL9920342 0.74 PDE4B (0.52) CSF1RPDE4BPDE4APDE4CPDE4D
SCHEMBL9920279 0.73 JAK1 (0.46) CSF1RTYK2
SCHEMBL1160264 0.72 JAK1 (0.65) TYK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120149691-A1 Pyrrolo [1,2-b] Pyridazine Derivatives as Janus Kinase Inhibitors BIOCRYST PHARMACEUTICALS, INC. (US) 2012-06-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120149691-A1 Pyrrolo [1,2-b] Pyridazine Derivatives as Janus Kinase Inhibitors JAK1, JAK2, JAK3 CSF1R 315/4885PDE4B 2524/4885PDE4A 2373/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.