SCHEMBL9923318

SCHEMBL9923318

Cc1cc2c(Oc3ccc(S(=O)(=O)N4CCC4)cc3)cc(C(=O)NC(=N)C=N)cc2o1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GCK P35557 7/20 0.51
KCNH2 Q12809 3/20 0.51
KMT2A Q03164 5/20 0.41
ALDH1A1 P00352 6/20 0.40
POLB P06746 2/20 0.39
HTT P42858 2/20 0.39
TSHR P16473 1/20 0.39
LMNA P02545 3/20 0.39
RXFP1 Q9HBX9 1/20 0.39
MAPT P10636 3/20 0.38
GAA P10253 2/20 0.38
RAB9A P51151 1/20 0.38
USP2 O75604 1/20 0.38
ALOX12 P18054 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2669336 0.90 GCK (0.47) GCKKCNH2KMT2AALDH1A1POLB
SCHEMBL643787 0.81 CYP2C9 (0.48) GCKKCNH2KMT2AALDH1A1POLB
SCHEMBL643930 0.80 GCK (0.58) GCKKCNH2
SCHEMBL645985 0.80 GCK (0.65) GCKKCNH2RXFP1
SCHEMBL642236 0.80 GCK (0.60) GCKKCNH2ALDH1A1POLBHTT
SCHEMBL643041 0.80 GCK (0.60) GCKKCNH2
SCHEMBL643556 0.79 GCK (0.63) GCKKCNH2KMT2AALDH1A1RXFP1
SCHEMBL643939 0.79 GCK (0.59) GCKKCNH2KMT2AALDH1A1MAPT
SCHEMBL644575 0.78 GCK (0.62) GCKKCNH2RXFP1MAPTRAB9A
SCHEMBL644391 0.78 GCK (0.67) GCKKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2463283-A1 Fused phenyl Amido heterocyclic compounds for the prevention and treatment of glucokinase-mediated diseases Pfizer Products Inc. (US) 2012-06-13 EP disclosed