SCHEMBL9928508

SCHEMBL9928508

CC#CCn1c(N2CCC[C@@H](N)C2)nc2[nH]c(=N)n(Cc3ccc(C#N)cc3)c(=O)c21

nearest known ligand 0.59

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 20/20 0.59
CHRM1 P11229 2/20 0.59
FAP Q12884 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3972634 0.85 DPP4 (0.80) DPP4CHRM1FAP
SCHEMBL3972638 0.85 DPP4 (0.80) DPP4CHRM1FAP
Hydrochloric Acid SCHEMBL2964308 0.83 DPP4 (0.58) DPP4CHRM1FAP
SCHEMBL3540700 0.81 DPP4 (0.65) DPP4CHRM1FAP
SCHEMBL3540704 0.81 DPP4 (0.65) DPP4CHRM1FAP
Hydrochloric Acid SCHEMBL2968054 0.81 DPP4 (0.62) DPP4CHRM1FAP
SCHEMBL3972106 0.77 DPP4 (0.74) DPP4CHRM1FAP
SCHEMBL3972113 0.77 DPP4 (0.74) DPP4CHRM1FAP
SCHEMBL3970600 0.77 DPP4 (0.75) DPP4CHRM1FAP
SCHEMBL3970592 0.77 DPP4 (0.75) DPP4CHRM1FAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2648517-B1 TRICYCLIC HETEROCYCLES USEFUL AS DIPEPTIDYL PEPTIDASE-IV INHIBITORS MERCK SHARP & DOHME (US) 2015-08-05 EP disclosed
WO-2012078448-A1 TRICYCLIC HETEROCYCLES USEFUL AS DIPEPTIDYL PEPTIDASE-IV INHIBITORS SCHERING CORPORATION (US) 2012-06-14 WO disclosed