SCHEMBL9936933

SCHEMBL9936933

COC(=O)c1c[nH]c2ncc(Cl)cc12

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AXL P30530 5/20 0.63
NR4A2 P43354 10/20 0.62
MAP2K1 Q02750 2/20 0.56
CREBBP Q92793 1/20 0.49
BRAF P15056 3/20 0.47
JAK2 O60674 1/20 0.46
BMPR1B O00238 1/20 0.45
PLK4 O00444 1/20 0.45
PIR O00625 1/20 0.45
AURKA O14965 1/20 0.45
DCLK1 O15075 1/20 0.45
EPHB6 O15197 1/20 0.45
RIPK2 O43353 1/20 0.45
STK16 O75716 1/20 0.45
OXSR1 O95747 1/20 0.45
MAP4K4 O95819 1/20 0.45
ABL1 P00519 1/20 0.45
RAF1 P04049 1/20 0.45
LCK P06239 1/20 0.45
FYN P06241 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17324586 0.84 BRAF (0.49) AXLNR4A2MAP2K1BRAFJAK2
SCHEMBL23412702 0.84 F7 (0.56) AXLNR4A2MAP2K1BRAFJAK2
SCHEMBL27795046 0.84 BRAF (0.54) AXLNR4A2MAP2K1BRAFJAK2
SCHEMBL9938466 0.83 AXL (0.64) AXLNR4A2MAP2K1CREBBPBRAF
SCHEMBL9938142 0.82 AXL (0.63) AXLNR4A2MAP2K1CREBBP
SCHEMBL30020999 0.82 AXL (0.63) AXLNR4A2MAP2K1CREBBP
SCHEMBL30676600 0.82 AXL (0.63) AXLNR4A2MAP2K1CREBBPBRAF
SCHEMBL1427263 0.82 AXL (0.63) AXLNR4A2MAP2K1CREBBPBRAF
SCHEMBL28489988 0.81 JAK2 (0.48) AXLNR4A2MAP2K1BRAFJAK2
SCHEMBL17321399 0.81 BRAF (0.47) AXLNR4A2MAP2K1BRAFJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250092036-A1 COMPOUNDS AND COMPOSITIONS FOR MODULATING THE ACTIVITY OF ERK NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, INC. 2025-03-20 US disclosed
WO-2025037229-A1 COMPOUNDS AND COMPOSITIONS FOR MODULATING THE ACTIVITY OF ERK NOVARTIS AG (CH) 2025-02-20 WO disclosed
US-8993523-B2 Dimeric IAP inhibitors NOVARTIS AG (CH) 2015-03-31 US disclosed
US-20130309247-A1 DIMERIC IAP INHIBITORS NOVARTIS AG (CH) 2013-11-21 US disclosed
EP-2651919-A1 DIMERIC IAP INHIBITORS Novartis AG (CH) 2013-10-23 EP disclosed
WO-2012080271-A1 DIMERIC IAP INHIBITORS NOVARTIS AG (CH) 2012-06-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130309247-A1 DIMERIC IAP INHIBITORS XIAP, BIRC5, BIRC2 AXL 4160/4885NR4A2 3995/4885MAP2K1 958/4885
US-20250092036-A1 COMPOUNDS AND COMPOSITIONS FOR MODULATING THE ACTIVITY OF ERK MAPK1, MAP3K1, MAPK6 AXL 2674/4885NR4A2 1975/4885MAP2K1 127/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.