SCHEMBL9940046

SCHEMBL9940046

O=C(O)C1CC(F)CN1C(=O)OCc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
POLB P06746 1/20 0.47
PSEN1 P49768 1/20 0.46
PSEN2 P49810 1/20 0.46
APH1B Q8WW43 1/20 0.46
NCSTN Q92542 1/20 0.46
APH1A Q96BI3 1/20 0.46
PSENEN Q9NZ42 1/20 0.46
AGTR2 P50052 2/20 0.46
HTR2C P28335 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
PDK1 Q15118 1/20 0.45
PDK2 Q15119 1/20 0.45
PDK3 Q15120 1/20 0.45
PDK4 Q16654 1/20 0.45
CYP2C19 P33261 1/20 0.44
ALDH1A1 P00352 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1150913 1.00 NPC1 (0.49) NPC1RAB9ASMN1; SMN2POLBPSEN1
SCHEMBL21874256 1.00 NPC1 (0.49) NPC1RAB9ASMN1; SMN2POLBPSEN1
SCHEMBL11450804 1.00 NPC1 (0.49) NPC1RAB9ASMN1; SMN2POLBPSEN1
SCHEMBL2499400 1.00 NPC1 (0.49) NPC1RAB9ASMN1; SMN2POLBPSEN1
SCHEMBL1334730 0.91 POLB (0.47) NPC1RAB9ASMN1; SMN2POLBPSEN1
SCHEMBL1335928 0.91 POLB (0.47) NPC1RAB9ASMN1; SMN2POLBPSEN1
SCHEMBL1335516 0.91 POLB (0.47) NPC1RAB9ASMN1; SMN2POLBPSEN1
SCHEMBL1335517 0.91 POLB (0.47) NPC1RAB9ASMN1; SMN2POLBPSEN1
SCHEMBL1335456 0.91 POLB (0.47) NPC1RAB9ASMN1; SMN2POLBPSEN1
SCHEMBL19540632 0.91 POLB (0.49) NPC1RAB9ASMN1; SMN2POLBPSEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4430035-A1 SELECT KRAS G12C INHIBITORS AND USES THEREOF 1200 Pharma LLC (US) 2024-09-18 EP disclosed
WO-2023086383-A1 SELECT KRAS G12C INHIBITORS AND USES THEREOF 1200 PHARMA LLC (US) 2023-05-19 WO disclosed
US-8203003-B2 4-fluoropyrrolidine-2-carbonyl fluoride compounds and their preparative methods UBE INDUSTRIES, LTD. (JP) 2012-06-19 US disclosed