SCHEMBL9941447

SCHEMBL9941447

Cc1ccc(C2=c3ccc4c5c(ccc4c3C=C2)=CC=CC5)nc1

nearest known ligand 0.34

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.34
CCR5 P51681 1/20 0.34
CCR8 P51685 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9941388 0.82 KDM4E (0.30) CCR1CCR5CCR8
SCHEMBL15903546 0.68
SCHEMBL29564692 0.68
SCHEMBL15903796 0.67
SCHEMBL14941252 0.61
SCHEMBL29447186 0.61
SCHEMBL18849413 0.59 CCR1 (0.50) CCR1CCR5CCR8HDAC6
SCHEMBL22224024 0.58 CCR1 (0.48) CCR1CCR5CCR8HDAC6
SCHEMBL9616686 0.58 CCR1 (0.48) CCR1CCR5CCR8HDAC6
SCHEMBL25860933 0.57 CCR1 (0.47) CCR1CCR5CCR8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2651916-A2 C-17-HETEROARYL STEROIDAL COMPOUNDS AS INHIBITORS OF CYP11B, CYP17, AND/OR CYP21 BioMarin Pharmaceutical Inc. (US) 2013-10-23 EP disclosed
WO-2012083112-A2 CYP11B, CYP17, AND/OR CYP21 INHIBITORS BIOMARIN PHARMACEUTICAL INC. (US) 2012-06-21 WO disclosed