SCHEMBL9942964

SCHEMBL9942964

Cc1cc(CNC(=O)c2nc3n(c(=O)c2O)CC2(CN)CCC3(NC(=O)C(=O)N(C)C)CC2)ccc1F

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.41
MMP13 P45452 10/20 0.36
KCNH2 Q12809 1/20 0.36
MMP10 P09238 5/20 0.35
MMP8 P22894 5/20 0.35
MMP9 P14780 1/20 0.32
KCNE1 P15382 1/20 0.31
CCR1 P32246 1/20 0.31
KCNQ1 P51787 1/20 0.31
SCD O00767 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9942940 0.94 CYP2C9 (0.39) CYP2C9MMP13KCNH2MMP10MMP8
SCHEMBL9905237 0.93 CYP2C9 (0.41) CYP2C9MMP13KCNH2MMP10MMP8
SCHEMBL9901023 0.93 CYP2C9 (0.41) CYP2C9MMP13KCNH2MMP10MMP8
SCHEMBL9942979 0.93 CYP2C9 (0.41) CYP2C9MMP13KCNH2MMP10MMP8
SCHEMBL9942909 0.93 CYP2C9 (0.41) CYP2C9MMP13KCNH2MMP10MMP8
SCHEMBL9904945 0.91 CYP2C9 (0.40) CYP2C9MMP13KCNH2MMP10MMP8
SCHEMBL9900910 0.91 CYP2C9 (0.42) CYP2C9MMP13KCNH2MMP10MMP8
SCHEMBL9943009 0.91 CYP2C9 (0.39) CYP2C9MMP13KCNH2MMP10MMP8
SCHEMBL16063234 0.91 CYP2C9 (0.39) CYP2C9MMP13KCNH2MMP10MMP8
SCHEMBL9900842 0.91 CYP2C9 (0.39) CYP2C9MMP13KCNH2MMP10MMP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012078834-A1 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-06-14 WO disclosed