SCHEMBL9942968

SCHEMBL9942968

Cc1cc(CNC(=O)c2nc3n(c(=O)c2O)CC2(CN)CCC3(N(C)C(=O)C(=O)N(C)C)CC2)ccc1F

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.43
MMP13 P45452 10/20 0.37
KCNH2 Q12809 1/20 0.37
MMP10 P09238 5/20 0.35
MMP8 P22894 5/20 0.35
SCD O00767 1/20 0.33
KCNE1 P15382 1/20 0.33
CCR1 P32246 1/20 0.33
KCNQ1 P51787 1/20 0.33
MMP9 P14780 1/20 0.32
WDR5 P61964 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9905123 0.93 CYP2C9 (0.43) CYP2C9MMP13KCNH2MMP10MMP8
SCHEMBL9901013 0.93 CYP2C9 (0.43) CYP2C9MMP13KCNH2MMP10MMP8
SCHEMBL9942952 0.93 CYP2C9 (0.43) CYP2C9MMP13KCNH2MMP10MMP8
SCHEMBL9905163 0.91 CYP2C9 (0.42) CYP2C9MMP13KCNH2MMP10MMP8
SCHEMBL9905194 0.91 CYP2C9 (0.41) CYP2C9MMP13KCNH2MMP10MMP8
SCHEMBL9901158 0.90 CYP2C9 (0.44) CYP2C9MMP13KCNH2MMP10MMP8
SCHEMBL9943015 0.90 CYP2C9 (0.44) CYP2C9MMP13KCNH2MMP10MMP8
SCHEMBL14234672 0.90 CYP2C9 (0.53) CYP2C9KCNH2SCDKCNE1CCR1
SCHEMBL9943088 0.90 CYP2C9 (0.46) CYP2C9MMP13KCNH2MMP10MMP8
SCHEMBL14212654 0.90 CYP2C9 (0.41) CYP2C9MMP13KCNH2MMP10MMP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012078834-A1 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-06-14 WO disclosed