SCHEMBL9943750

SCHEMBL9943750

CC(C)[C@@H](C(=O)NC(Cc1ccccc1)CC(O)C(Cc1ccccc1)OC(N)=O)N1CCCNC1=O

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.64
ABCC3 O15438 1/20 0.64
ABCC4 O15439 1/20 0.64
ABCB11 O95342 1/20 0.64
PGR P06401 1/20 0.64
ABCB1 P08183 1/20 0.64
ADORA3 P0DMS8 1/20 0.64
CHRM1 P11229 1/20 0.64
TBXA2R P21731 1/20 0.64
ADRA1A P35348 1/20 0.64
OPRM1 P35372 1/20 0.64
HTR2B P41595 1/20 0.64
KCNH2 Q12809 1/20 0.64
SCN5A Q14524 1/20 0.64
ABCG2 Q9UNQ0 1/20 0.64
CA2 P00918 1/20 0.36
SDCBP O00560 2/20 0.36
SDC2 P34741 2/20 0.36
REN P00797 3/20 0.35
CTSD P07339 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9943748 1.00 CYP3A4 (0.64) CYP3A4ABCC3ABCC4ABCB11PGR
SCHEMBL9943746 1.00 CYP3A4 (0.64) CYP3A4ABCC3ABCC4ABCB11PGR
SCHEMBL9943725 0.84 CYP3A4 (0.77) CYP3A4ABCC3ABCC4ABCB11PGR
SCHEMBL9943595 0.84 CYP3A4 (0.77) CYP3A4ABCC3ABCC4ABCB11PGR
SCHEMBL4245489 0.84 CYP3A4 (0.77) CYP3A4ABCC3ABCC4ABCB11PGR
SCHEMBL9943769 0.83 CYP3A4 (0.54) CYP3A4ABCC3ABCC4ABCB11PGR
SCHEMBL9943771 0.83 CYP3A4 (0.54) CYP3A4ABCC3ABCC4ABCB11PGR
SCHEMBL21425157 0.83 CYP3A4 (0.63) CYP3A4ABCC3ABCC4ABCB11PGR
SCHEMBL4174124 0.83 CYP3A4 (0.60) CYP3A4ABCC3ABCC4ABCB11PGR
SCHEMBL5385947 0.81 CYP3A4 (0.59) CYP3A4ABCC3ABCC4ABCB11PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2465856-A2 Cytochrome P450 oxidase inhibitors and uses thereof Abbott Laboratories (US) 2012-06-20 EP disclosed