SCHEMBL9947627

SCHEMBL9947627

CCCOc1c2c(c(OCc3ccccc3)c3ccccc13)C(=O)N(c1ccc(CC(=O)O)cc1F)C2=O

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 16/20 0.57
CYP1A2 P05177 1/20 0.53
CYP2D6 P10635 1/20 0.53
PTGDR2 Q9Y5Y4 1/20 0.41
BRD4 O60885 1/20 0.36
USP2 O75604 1/20 0.36
ALDH1A1 P00352 1/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2298118 0.95 PTGER4 (0.61) PTGER4CYP1A2CYP2D6PTGDR2ALDH1A1
SCHEMBL9947691 0.93 PTGER4 (0.58) PTGER4CYP1A2CYP2D6PTGDR2BRD4
SCHEMBL2929004 0.92 PTGER4 (0.66) PTGER4CYP1A2CYP2D6PTGDR2
SCHEMBL10058518 0.91 PTGER4 (0.49) PTGER4CYP1A2CYP2D6PTGDR2ALDH1A1
SCHEMBL9947684 0.91 PTGER4 (0.57) PTGER4CYP1A2CYP2D6PTGDR2ALDH1A1
SCHEMBL13177214 0.90 PTGER4 (0.54) PTGER4CYP1A2CYP2D6PTGDR2BRD4
SCHEMBL1590037 0.89 PTGER4 (0.55) PTGER4CYP1A2CYP2D6PTGDR2
SCHEMBL9947708 0.89 PTGER4 (0.57) PTGER4CYP1A2CYP2D6PTGDR2BRD4
SCHEMBL9947668 0.88 PTGER4 (0.54) PTGER4CYP1A2CYP2D6PTGDR2
SCHEMBL10079536 0.88 PTGER4 (0.42) PTGER4CYP1A2CYP2D6USP2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8207213-B2 Benzoisoindole derivatives for the treatment of pain GLAXO GROUP LIMITED (GB) 2012-06-26 US disclosed