SCHEMBL9947702

SCHEMBL9947702

CC(C)Oc1c2c(c(OCc3ccccc3)c3ccccc13)C(=O)N(c1ccc(CC(=O)O)cc1Cl)C2=O

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 15/20 0.54
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
EDNRA P25101 1/20 0.38
GLRA1 P23415 1/20 0.37
BRD4 O60885 1/20 0.36
USP2 O75604 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.35
HSD17B10 Q99714 1/20 0.35
PPARD Q03181 1/20 0.35
NR1H4 Q96RI1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2926013 0.93 PTGER4 (0.55) PTGER4CYP1A2CYP2D6ALDH1A1HSD17B10
SCHEMBL2936637 0.92 PTGER4 (0.58) PTGER4CYP1A2CYP2D6BRD4USP2
SCHEMBL10058525 0.90 PTGER4 (0.48) PTGER4CYP1A2CYP2D6EDNRAALDH1A1
SCHEMBL9948014 0.90 PTGER4 (0.66) PTGER4CYP1A2CYP2D6
SCHEMBL9947668 0.89 PTGER4 (0.54) PTGER4CYP1A2CYP2D6EDNRA
SCHEMBL1590841 0.89 PTGER4 (0.51) PTGER4CYP1A2CYP2D6ALDH1A1HSD17B10
SCHEMBL9947978 0.89 PTGER4 (0.51) PTGER4CYP1A2CYP2D6ALDH1A1HSD17B10
SCHEMBL9947708 0.88 PTGER4 (0.57) PTGER4CYP1A2CYP2D6BRD4USP2
SCHEMBL11967825 0.86 EDNRA (0.41) PTGER4CYP1A2CYP2D6EDNRAGLRA1
SCHEMBL4410567 0.84 PTGER4 (0.69) PTGER4CYP1A2CYP2D6EDNRAUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8207213-B2 Benzoisoindole derivatives for the treatment of pain GLAXO GROUP LIMITED (GB) 2012-06-26 US disclosed