SCHEMBL9947762

SCHEMBL9947762

CCOc1c2c(c(OCc3ccccc3)c3ccccc13)C(=O)N(c1ccc(CC(=O)O)c(F)c1)C2=O

nearest known ligand 0.67

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 20/20 0.67
CYP1A2 P05177 1/20 0.64
CYP2D6 P10635 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9947957 0.95 PTGER4 (0.59) PTGER4CYP1A2CYP2D6
SCHEMBL4611730 0.94 PTGER4 (0.74) PTGER4CYP1A2CYP2D6
SCHEMBL9947679 0.93 PTGER4 (0.58) PTGER4CYP1A2CYP2D6
SCHEMBL10058524 0.92 PTGER4 (0.57) PTGER4CYP1A2CYP2D6
SCHEMBL9947630 0.90 PTGER4 (0.54) PTGER4CYP1A2CYP2D6
SCHEMBL10058498 0.90 PTGER4 (0.54) PTGER4CYP1A2CYP2D6
SCHEMBL9947656 0.89 PTGER4 (0.68) PTGER4CYP1A2CYP2D6
SCHEMBL1590148 0.88 PTGER4 (0.66) PTGER4CYP1A2CYP2D6
SCHEMBL10078913 0.86 PTGER4 (0.51) PTGER4CYP1A2CYP2D6
SCHEMBL8588489 0.86 PTGER4 (0.63) PTGER4CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979317-B1 BENZOISOINDOLE DERIVATIVES FOR THE TREATMENT OF PAIN GLAXO GROUP LTD (GB) 2012-08-22 EP disclosed
US-8207213-B2 Benzoisoindole derivatives for the treatment of pain GLAXO GROUP LIMITED (GB) 2012-06-26 US disclosed