SCHEMBL9952486

SCHEMBL9952486

NC(=O)Nc1ccc(NCc2ccc(F)cc2)nc1N

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNQ3 O43525 3/20 0.70
KCNQ2 O43526 3/20 0.70
ABCB11 O95342 1/20 0.70
ESR1 P03372 1/20 0.70
CYP1A2 P05177 1/20 0.70
CYP3A4 P08684 1/20 0.70
HTR1A P08908 1/20 0.70
ADRA2A P08913 1/20 0.70
ADORA3 P0DMS8 1/20 0.70
CYP2D6 P10635 1/20 0.70
CYP2C9 P11712 1/20 0.70
ALOX15 P16050 1/20 0.70
NFKB1 P19838 1/20 0.70
TBXA2R P21731 1/20 0.70
MAPK1 P28482 1/20 0.70
CASP1 P29466 1/20 0.70
CYP2C19 P33261 1/20 0.70
SHMT2 P34897 1/20 0.70
PTGS2 P35354 1/20 0.70
OPRK1 P41145 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12505604 0.89 KCNQ3 (0.74) KCNQ3KCNQ2ABCB11ESR1CYP1A2
SCHEMBL4890687 0.88 KCNQ3 (0.72) KCNQ3KCNQ2ABCB11ESR1CYP1A2
Hydrochloric Acid SCHEMBL31741641 0.87 KCNQ3 (0.71) KCNQ3KCNQ2ABCB11ESR1CYP1A2
Hydrochloric Acid SCHEMBL10786035 0.87 KCNQ3 (0.71) KCNQ3KCNQ2ABCB11ESR1CYP1A2
SCHEMBL20641737 0.86 KCNQ3 (0.80) KCNQ3KCNQ2ABCB11ESR1CYP1A2
SCHEMBL29754330 0.83 KCNQ3 (0.69) KCNQ3KCNQ2ABCB11ESR1CYP1A2
SCHEMBL10786711 0.83 KCNQ3 (0.69) KCNQ3KCNQ2ABCB11ESR1CYP1A2
Flupirtine SCHEMBL25009 0.83 KCNQ2 (1.00) KCNQ3KCNQ2ABCB11ESR1CYP1A2
SCHEMBL20654773 0.83 KCNQ3 (0.76) KCNQ3KCNQ2ABCB11ESR1CYP1A2
Flupirtine SCHEMBL15357226 0.83 KCNQ2 (1.00) KCNQ3KCNQ2ABCB11ESR1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2655328-A1 NOVEL MULTICOMPONENT CRYSTALS MADE OF ([2-AMINO-6-(4-FLUORO-BENZYLAMINO)- PYRIDIN-3-YL]-CARBAMIC ACID ETHYL ESTER AND 2-[2-[(2,6-DICHLORPHENYL)-AMINO]-PHENYL]-ACETIC ACID AWD.pharma GmbH & Co.KG (DE) 2013-10-30 EP disclosed
WO-2012084975-A1 NOVEL MULTICOMPONENT CRYSTALS MADE OF ([2-AMINO-6-(4-FLUORO-BENZYLAMINO)- PYRIDIN-3-YL]-CARBAMIC ACID ETHYL ESTER AND 2-[2-[(2,6-DICHLORPHENYL)-AMINO]-PHENYL]-ACETIC ACID AWD.PHARMA GMBH & CO. KG (DE) 2012-06-28 WO disclosed