SCHEMBL9953073

SCHEMBL9953073

Cc1ccc2c(c1)c(I)nn2C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ELANE P08246 6/20 0.40
POLB P06746 4/20 0.40
KDM4E B2RXH2 3/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
HSD17B10 Q99714 1/20 0.40
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
MAPT P10636 2/20 0.37
THRB P10828 1/20 0.37
HPGD P15428 1/20 0.37
RAB9A P51151 1/20 0.37
LMNA P02545 1/20 0.36
ALDH1A1 P00352 1/20 0.35
MARK4 Q96L34 1/20 0.35
APEX1 P27695 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
DAO P14920 2/20 0.35
NR1I2 O75469 1/20 0.35
AHR P35869 1/20 0.35
PDE5A O76074 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14739013 0.82 ELANE (0.36) ELANEPOLBKDM4EHSD17B10MAPT
SCHEMBL3636090 0.81 ELANE (0.45) ELANEL3MBTL1MEN1KMT2ALMNA
SCHEMBL3518728 0.81 CHEK1 (0.39) ELANEPOLBKDM4EHSD17B10MEN1
SCHEMBL9952523 0.80 MAP2K4 (0.42) ELANEPOLBKDM4EL3MBTL1HSD17B10
SCHEMBL14631678 0.78 PTGDR2 (0.46) POLBKDM4EL3MBTL1HSD17B10MAPT
SCHEMBL9952327 0.76 ELANE (0.45) ELANEPOLBKDM4EHSD17B10F2
SCHEMBL3518373 0.76 ELANE (0.50) ELANEL3MBTL1MEN1KMT2AMAPT
SCHEMBL14738967 0.75 CPT1A (0.36) ELANEPOLBMEN1KMT2AMAPT
SCHEMBL15792144 0.74 ADORA2A (0.39) POLBKDM4EL3MBTL1HSD17B10MEN1
SCHEMBL14738410 0.74 CA12 (0.41) ELANEKDM4EHSD17B10HPGDRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2655357-A1 INDAZOLYL TRIAZOLE DERIVATIVES AS IRAK INHIBITORS Merck Serono S.A. (CH) 2013-10-30 EP disclosed
WO-2012084704-A1 INDAZOLYL TRIAZOLE DERIVATIVES AS IRAK INHIBITORS MERCK SERONO S.A. (CH) 2012-06-28 WO disclosed