SCHEMBL9954399

SCHEMBL9954399

COC(=O)c1c(-c2ccc(F)cc2)oc2cc(N)c(OC(C)C)cc12.COC(=O)c1c(-c2ccc(F)cc2)oc2cc(NS(C)(=O)=O)c(OC(C)C)cc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
IKBKB O14920 1/20 0.35
RCE1 Q9Y256 1/20 0.35
LMNA P02545 2/20 0.35
CYP19A1 P11511 1/20 0.34
ANO1 Q5XXA6 2/20 0.34
BRD4 O60885 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
MAPT P10636 3/20 0.33
TP53 P04637 2/20 0.33
PIK3CA P42336 1/20 0.33
F11 P03951 1/20 0.33
F2 P00734 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ACLY P53396 1/20 0.32
HPGD P15428 1/20 0.32
ALDH1A1 P00352 1/20 0.32
PTGS2 P35354 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1918337 0.95 ATM (0.40) ATML3MBTL1RCE1LMNACYP19A1
SCHEMBL2297611 0.90 ATM (0.43) ATML3MBTL1IKBKBRCE1LMNA
SCHEMBL1919350 0.87 KDM4E (0.39) LMNACYP19A1ANO1F2KDM4E
SCHEMBL1919537 0.86 ANO1 (0.43) CYP19A1ANO1MEN1KMT2AKDM4E
SCHEMBL3533863 0.86 KDM4E (0.47) L3MBTL1RCE1MEN1KMT2AMAPT
SCHEMBL2363613 0.85 CYP2C9 (0.43)
SCHEMBL2844773 0.85 CYP19A1 (0.37) CYP19A1ANO1ALDH1A1PTGS2
SCHEMBL1918630 0.85 CYP19A1 (0.37) CYP19A1ANO1F2ACLYPTGS2
SCHEMBL29950180 0.85 CYP2C9 (0.43)
SCHEMBL2835706 0.82 CYP3A4 (0.36) CYP19A1ANO1F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2655362-A1 HEPATITIS C INHIBITORS AND USES THEREOF Abbvie Inc. (US) 2013-10-30 EP disclosed
WO-2012087833-A1 HEPATITIS C INHIBITORS AND USES THEREOF ABBOTT LABORATORIES (US) 2012-06-28 WO disclosed