SCHEMBL9957044

SCHEMBL9957044

Cc1ccc(-n2nccn2)c(C=O)c1N1C[C@H]2CCN(c3nc4ccc(F)cc4s3)C[C@H]21

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 17/20 0.43
HCRTR2 O43614 17/20 0.43
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
ALDH1A1 P00352 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9957138 0.83 HCRTR1 (0.50) HCRTR1HCRTR2
SCHEMBL9954554 0.80 HCRTR1 (0.54) HCRTR1HCRTR2
SCHEMBL9955934 0.78 HCRTR1 (0.48) HCRTR1HCRTR2
SCHEMBL9957650 0.78 HCRTR1 (0.56) HCRTR1HCRTR2LMNATP53
SCHEMBL9957647 0.78 HCRTR1 (0.56) HCRTR1HCRTR2LMNATP53
SCHEMBL9957155 0.77 HCRTR1 (0.41) HCRTR1HCRTR2
SCHEMBL9954517 0.77 HCRTR1 (0.41) HCRTR1HCRTR2
SCHEMBL9957391 0.77 HCRTR1 (0.41) HCRTR1HCRTR2
SCHEMBL9956933 0.76 HCRTR1 (0.41) HCRTR1HCRTR2
SCHEMBL9957419 0.76 HCRTR1 (0.42) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085852-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-8-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO claimed
WO-2012085852-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-8-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed