SCHEMBL9957367

SCHEMBL9957367

Cc1ccc(-n2cccn2)c(C(=O)N2C[C@H]3CCN(c4cnc5cc(F)ccc5n4)C[C@H]32)c1F

nearest known ligand 0.47

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 17/20 0.47
HCRTR1 O43613 16/20 0.47
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9957079 0.89 HCRTR1 (0.57) HCRTR2HCRTR1
SCHEMBL9956544 0.89 HCRTR1 (0.57) HCRTR2HCRTR1
SCHEMBL9957552 0.89 HCRTR1 (0.57) HCRTR2HCRTR1
SCHEMBL9957554 0.89 HCRTR1 (0.57) HCRTR2HCRTR1
SCHEMBL9957704 0.89 HCRTR2 (0.52) HCRTR2HCRTR1
SCHEMBL9957269 0.87 HCRTR2 (0.41) HCRTR2HCRTR1CYP3A4
SCHEMBL9955407 0.86 HCRTR1 (0.59) HCRTR2HCRTR1
SCHEMBL9954146 0.86 HCRTR1 (0.59) HCRTR2HCRTR1
SCHEMBL9955441 0.86 HCRTR1 (0.59) HCRTR2HCRTR1
SCHEMBL9957037 0.83 HCRTR1 (0.45) HCRTR2HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085852-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-8-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed