SCHEMBL9957712

SCHEMBL9957712

Cc1ccc(-n2nccn2)c(C(=O)N2CC3CCN(C(=O)O)CC32)c1F

nearest known ligand 0.49

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 20/20 0.49
HCRTR2 O43614 20/20 0.49
CYP3A4 P08684 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9955951 0.92 HCRTR1 (0.54) HCRTR1HCRTR2
SCHEMBL14973561 0.84 HCRTR1 (0.63) HCRTR1HCRTR2
SCHEMBL9960725 0.83 HCRTR1 (0.49) HCRTR1HCRTR2
SCHEMBL9956100 0.83 HCRTR1 (0.49) HCRTR1HCRTR2
Hydrochloric Acid SCHEMBL9957524 0.82 HCRTR1 (0.47) HCRTR1HCRTR2CYP3A4
Hydrochloric Acid SCHEMBL9957521 0.82 HCRTR1 (0.47) HCRTR1HCRTR2CYP3A4
SCHEMBL9957016 0.80 HCRTR2 (0.65) HCRTR1HCRTR2
SCHEMBL9955630 0.79 HCRTR1 (0.47) HCRTR1HCRTR2CYP3A4
SCHEMBL9957554 0.77 HCRTR1 (0.57) HCRTR1HCRTR2
SCHEMBL9957079 0.77 HCRTR1 (0.57) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085852-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-8-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed