SCHEMBL9974994

SCHEMBL9974994

c1cncc(-c2cc(-c3cccnc3)c(-c3ccc(-c4cnccn4)cc3)cc2-c2ccc(-c3cnccn3)cc2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 7/20 0.49
ALDH1A1 P00352 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
MKNK1 Q9BUB5 1/20 0.46
MKNK2 Q9HBH9 1/20 0.46
PIM2 Q9P1W9 1/20 0.44
CYP19A1 P11511 3/20 0.44
CYP2C9 P11712 2/20 0.44
CYP2C19 P33261 2/20 0.44
CYP2D6 P10635 1/20 0.44
LOXL2 Q9Y4K0 1/20 0.44
NUDT1 P36639 1/20 0.44
CYP11B1 P15538 3/20 0.44
PIK3CA P42336 1/20 0.43
KMO O15229 2/20 0.43
PTGS2 P35354 1/20 0.43
CHEK2 O96017 1/20 0.43
CYP11B2 P19099 2/20 0.42
CYP2E1 P05181 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9974960 0.95 CYP2A6 (0.50) CYP2A6ALDH1A1CYP1A2CYP3A4MKNK1
SCHEMBL9974946 0.89 PIM1 (0.48) CYP2A6ALDH1A1PIM2CYP19A1CYP2C9
SCHEMBL9974997 0.88 PIM1 (0.47) CYP2A6ALDH1A1PIM2CYP19A1CYP2C9
SCHEMBL9974928 0.85 CYP2A6 (0.71) CYP2A6ALDH1A1CYP1A2CYP3A4MKNK1
SCHEMBL4672073 0.83 CYP2A6 (0.67) CYP2A6ALDH1A1CYP1A2CYP3A4MKNK1
SCHEMBL31140239 0.83 CYP2A6 (0.67) CYP2A6ALDH1A1CYP1A2CYP3A4MKNK1
SCHEMBL9974932 0.83 CYP2A6 (0.53) CYP2A6CYP1A2CYP3A4CYP19A1CYP2C9
SCHEMBL9974953 0.82 CYP2D6 (0.46) PIM2CYP19A1CYP2C9CYP2C19CYP2D6
SCHEMBL9974998 0.82 PIM2 (0.45) CYP2A6PIM2CYP19A1CYP2C9CYP2C19
SCHEMBL9975001 0.81 CYP2A6 (0.47) CYP2A6CYP1A2CYP19A1CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012081541-A1 1, 2, 4, 5-SUBSTITUTED PHENYL DERIVATIVE, PRODUCTION METHOD FOR SAME, AND ORGANIC ELECTROLUMINESCENT ELEMENT 東ソー株式会社 (JP) 2012-06-21 WO disclosed