SCHEMBL9975856

SCHEMBL9975856

CC1CCC(C2=C(c3cc(C#CC(C)(C)C)sc3C(N)=O)CN(CC3CCOCC3)CC2)CC1

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP2E1 P05181 1/20 0.41
NR1I2 O75469 2/20 0.36
GRM2 Q14416 2/20 0.32
C5AR1 P21730 1/20 0.32
OPRM1 P35372 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10324617 0.93 CYP2E1 (0.47) CYP2E1NR1I2
SCHEMBL10324262 0.88 CYP2E1 (0.44) CYP2E1NR1I2C5AR1
SCHEMBL10366310 0.86 CYP2E1 (0.38) CYP2E1NR1I2C5AR1
SCHEMBL9975906 0.82 CYP2E1 (0.43) CYP2E1NR1I2
SCHEMBL10381443 0.79 CYP2E1 (0.33) CYP2E1
SCHEMBL9976063 0.79 NR1I2 (0.45) CYP2E1NR1I2
SCHEMBL19402939 0.78 CYP2E1 (0.32) CYP2E1C5AR1
SCHEMBL9975843 0.78 NR1I2 (0.44) CYP2E1NR1I2
SCHEMBL9975886 0.78 NR1I2 (0.44) CYP2E1NR1I2
SCHEMBL9975799 0.77 NR1I2 (0.43) CYP2E1NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012083105-A1 INHIBITORS OF HEPATITIS C VIRUS POLYMERASE COCRYSTAL DISCOVERY, INC. (US) 2012-06-21 WO disclosed