SCHEMBL9975896

SCHEMBL9975896

COC(=O)c1sc(-c2ccc(NC(=O)c3cscn3)cc2)cc1C1=C(C2CCC(C)CC2)CNCC1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 4/20 0.35
GRM4 Q14833 2/20 0.35
MAPT P10636 3/20 0.33
ROCK2 O75116 1/20 0.33
TP53 P04637 1/20 0.33
KDM4E B2RXH2 2/20 0.32
RXFP1 Q9HBX9 1/20 0.32
HTT P42858 1/20 0.32
ATM Q13315 1/20 0.32
GRM1 Q13255 1/20 0.32
PARP1 P09874 1/20 0.32
STAT1 P42224 1/20 0.31
NPC1 O15118 1/20 0.31
CASP3 P42574 1/20 0.31
RAB9A P51151 1/20 0.31
SENP8 Q96LD8 1/20 0.31
SENP7 Q9BQF6 1/20 0.31
SENP6 Q9GZR1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10324943 0.93 GRM4 (0.34) GRM4ROCK2GRM1PARP1
SCHEMBL10325384 0.86 NAMPT (0.35) PTPN1GRM4MAPTROCK2TP53
SCHEMBL9941709 0.81 KDM4E (0.46) MAPTTP53KDM4EHTTATM
SCHEMBL10325054 0.80 KMT2A (0.35) GRM4MAPTTP53KDM4ERXFP1
SCHEMBL10365294 0.80 NAMPT (0.36) GRM4ROCK2
SCHEMBL16866379 0.79 NAMPT (0.35) PTPN1GRM4MAPTROCK2TP53
SCHEMBL10366103 0.79 NAMPT (0.35) GRM4ROCK2GRM1
SCHEMBL10324459 0.79 NAMPT (0.35) GRM4ROCK2GRM1
SCHEMBL10324542 0.79 NAMPT (0.35) PTPN1GRM4MAPTROCK2TP53
SCHEMBL10324335 0.79 NAMPT (0.32) GRM4ROCK2GRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012083105-A1 INHIBITORS OF HEPATITIS C VIRUS POLYMERASE COCRYSTAL DISCOVERY, INC. (US) 2012-06-21 WO disclosed