SCHEMBL997620

SCHEMBL997620

O=CC(Oc1ccccc1)N1CCn2c(nc(-c3ccc(F)cc3)c2Nc2ccc(Cl)c(F)c2)C1

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 14/20 0.57
CYP3A4 P08684 1/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
CSNK1D P48730 1/20 0.30
MAPK14 Q16539 1/20 0.30
KDM4E B2RXH2 1/20 0.30
USP2 O75604 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
GAA P10253 1/20 0.30
HPGD P15428 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL997258 0.84 KCNH2 (0.65) KCNH2CYP3A4
SCHEMBL999114 0.78 KCNH2 (0.59) KCNH2CYP3A4
SCHEMBL997618 0.78 KCNH2 (0.75) KCNH2CYP3A4POLBMAPTUSP2
SCHEMBL997952 0.76 KCNH2 (0.63) KCNH2CYP3A4CSNK1DKDM4EUSP2
SCHEMBL2069847 0.75 KCNH2 (0.79) KCNH2CYP3A4CSNK1D
SCHEMBL997524 0.75 KCNH2 (0.61) KCNH2CYP3A4KDM4EUSP2ALDH1A1
SCHEMBL997860 0.74 KCNH2 (0.58) KCNH2CYP3A4PTGDR2
SCHEMBL12952283 0.74 KCNH2 (0.75) KCNH2CYP3A4CSNK1D
SCHEMBL997932 0.74 KCNH2 (0.63) KCNH2CYP3A4CSNK1DKDM4EUSP2
SCHEMBL2069915 0.74 KCNH2 (0.69) KCNH2CYP3A4CSNK1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2451814-A2 FUSED IMIDAZOLES AND COMPOSITIONS COMPRISING THEM FOR THE TREATMENT OF PARASITIC DISEASES, SUCH AS E.G. MALARIA IRM LLC (BM) 2012-05-16 EP claimed
WO-2011006143-A2 COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF PARASITIC DISEASES IRM LLC (BM) 2011-01-13 WO claimed