SCHEMBL9977889

SCHEMBL9977889

Cc1ccc(N2N=CCN2)c(C(=O)NCCn2ccc(-c3cccc(C)n3)n2)c1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 5/20 0.49
HCRTR2 O43614 5/20 0.49
PDE10A Q9Y233 1/20 0.34
TGFBR1 P36897 6/20 0.34
TGFBR2 P37173 4/20 0.34
DRD2 P14416 3/20 0.34
DRD4 P21917 3/20 0.34
HTR1A P08908 2/20 0.34
AR P10275 1/20 0.33
NAMPT P43490 1/20 0.33
GRM5 P41594 1/20 0.32
KDM5B Q9UGL1 1/20 0.32
DRD3 P35462 1/20 0.32
SORT1 Q99523 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15326992 0.83 HCRTR1 (0.69) HCRTR1HCRTR2
SCHEMBL9977862 0.67 HCRTR1 (0.71) HCRTR1HCRTR2
SCHEMBL9977850 0.66 HCRTR1 (0.79) HCRTR1HCRTR2
SCHEMBL29839048 0.64 CCR1 (0.50) TGFBR1TGFBR2GRM5
SCHEMBL9977796 0.63 HCRTR1 (0.74) HCRTR1HCRTR2
SCHEMBL15338621 0.62 HCRTR1 (0.58) HCRTR1HCRTR2PDE10AAR
SCHEMBL9977902 0.62 HCRTR1 (0.72) HCRTR1HCRTR2
SCHEMBL9977852 0.62 CCR1 (0.50) TGFBR1TGFBR2
SCHEMBL15604615 0.61 HCRTR1 (0.50) HCRTR1HCRTR2NAMPT
SCHEMBL15604579 0.59 HCRTR1 (0.49) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012081692-A1 PYRAZOLE DERIVATIVE 大正製薬株式会社 (JP) 2012-06-21 WO disclosed