SCHEMBL9978159

SCHEMBL9978159

CC(=O)c1ccc(OCC(F)(F)F)c(-c2ccc(Cl)cc2)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.42
CNR2 P34972 1/20 0.42
CTSA P10619 5/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.39
MRGPRX4 Q96LA9 2/20 0.39
MAPT P10636 3/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
KCNK3 O14649 1/20 0.38
KCNK9 Q9NPC2 1/20 0.38
FFAR4 Q5NUL3 3/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
RXFP1 Q9HBX9 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
RECQL P46063 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL410512 0.89 MRGPRX4 (0.49) CNR1CNR2CTSAPTGDR2MRGPRX4
SCHEMBL411012 0.88 MRGPRX4 (0.52) CNR1CNR2CTSAMRGPRX4MAPT
SCHEMBL31267243 0.80 CNR1 (0.45) CNR1CNR2CTSAMAPTMEN1
SCHEMBL21634885 0.80 CNR1 (0.45) CNR1CNR2CTSAMAPTMEN1
SCHEMBL411488 0.80 KDM4E (0.37) CNR1CNR2PTGDR2MAPTKCNK3
SCHEMBL9935119 0.78 CTSA (0.41) CNR1CNR2CTSAMRGPRX4MAPT
SCHEMBL9978011 0.77 PTGDR2 (0.46) CNR1CNR2PTGDR2MAPTMEN1
SCHEMBL21634717 0.76 TTR (0.47) MRGPRX4MAPTMEN1KMT2A
SCHEMBL31267253 0.76 TTR (0.47) MRGPRX4MAPTMEN1KMT2A
SCHEMBL21634704 0.75 NOTUM (0.46) CNR2CTSAMRGPRX4MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012080144-A1 OXIME COMPOUNDS AS HDL-CHOLESTEROL RAISING AGENTS F. HOFFMANN-LA ROCHE AG (CH) 2012-06-21 WO disclosed