SCHEMBL9979744

SCHEMBL9979744

NS(=O)(=O)c1ccc(-n2nc(CCCNC(=O)I)cc2-c2ccccc2)cc1

nearest known ligand 0.78

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 15/20 0.78
PTGS2 P35354 14/20 0.71
CA1 P00915 3/20 0.69
CA2 P00918 3/20 0.69
CA9 Q16790 3/20 0.69
AKR1C3 P42330 1/20 0.68
PTGS1 P23219 4/20 0.61
ALOX5 P09917 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24398220 0.91 EPHX2 (0.79) EPHX2PTGS2CA1CA2CA9
SCHEMBL9937759 0.87 EPHX2 (1.00) EPHX2PTGS2CA1CA2CA9
SCHEMBL15460602 0.85 EPHX2 (0.71) EPHX2PTGS2CA1CA2CA9
SCHEMBL3248374 0.84 CA1 (0.87) EPHX2PTGS2CA1CA2CA9
SCHEMBL15460598 0.84 EPHX2 (0.88) EPHX2PTGS2CA1CA2CA9
SCHEMBL9938576 0.84 EPHX2 (1.00) EPHX2PTGS2CA1CA2CA9
SCHEMBL9938872 0.84 EPHX2 (0.80) EPHX2PTGS2CA1CA2CA9
SCHEMBL15455650 0.83 CA1 (0.77) EPHX2PTGS2CA1CA2CA9
SCHEMBL9938352 0.83 EPHX2 (1.00) EPHX2PTGS2CA1CA2CA9
SCHEMBL15460596 0.82 EPHX2 (0.85) EPHX2PTGS2CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012082647-A2 PYRAZOLE INHIBITORS OF COX-2 AND sEH THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2012-06-21 WO disclosed