SCHEMBL9987461

SCHEMBL9987461

CC(COCc1ccccc1)Oc1cc(Oc2ccc(S(C)(=O)=O)cc2)cc(C(=N)N)c1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GCK P35557 19/20 0.47
KCNH2 Q12809 3/20 0.45
PRSS1 P07477 1/20 0.40
PRSS2 P07478 1/20 0.40
PRSS3 P35030 1/20 0.40
ST14 Q9Y5Y6 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9987460 1.00 GCK (0.47) GCKKCNH2PRSS1PRSS2PRSS3
SCHEMBL3598462 0.89 GCK (0.55) GCKKCNH2
SCHEMBL2664229 0.88 GCK (0.50) GCKKCNH2
SCHEMBL12070254 0.87 GCK (0.44) GCKKCNH2
SCHEMBL2664227 0.86 GCK (0.53) GCKKCNH2
SCHEMBL9986858 0.85 GCK (0.45) GCKKCNH2
SCHEMBL3595253 0.85 GCK (0.45) GCKKCNH2
SCHEMBL9986959 0.85 GCK (0.59) GCKKCNH2
SCHEMBL9986958 0.85 GCK (0.59) GCKKCNH2
SCHEMBL9071277 0.82 GCK (0.56) GCKKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011158149-A1 2-(3,5-DISUBSTITUTEDPHENYL)PYRIMIDIN-4(3H)-ONE DERIVATIVES PFIZER INC. (US) 2011-12-22 WO disclosed