Benzo[E]Pyrene

Benzo[E]Pyrene

SCHEMBL9998154

c1ccc2c(c1)c1cccc3ccc4cccc2c4c31.c1ccc2c(c1)ccc1c2ccc2c3ccccc3ccc21

nearest known ligand 0.84

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 7/20 0.84
ALDH1A1 P00352 6/20 0.84
HPGD P15428 5/20 0.84
CYP1A2 P05177 3/20 0.84
THRB P10828 1/20 0.84
HPRT1 P00492 3/20 0.74
ERBB2 P04626 1/20 0.71
FYN P06241 1/20 0.71
MAOA P21397 1/20 0.71
ACHE P22303 1/20 0.71
AHR P35869 1/20 0.71
TSHR P16473 5/20 0.63
TDP1 Q9NUW8 3/20 0.63
CYP2A6 P11509 1/20 0.63
HIF1A Q16665 3/20 0.52
CYP1B1 Q16678 2/20 0.52
PAX8 Q06710 1/20 0.52
CYP3A4 P08684 4/20 0.50
L3MBTL1 Q9Y468 3/20 0.50
CYP1A1 P04798 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4854359 0.95 HSD17B10 (0.76) HSD17B10ALDH1A1HPGDCYP1A2THRB
SCHEMBL29578620 0.95 HSD17B10 (0.76) HSD17B10ALDH1A1HPGDCYP1A2THRB
Chrysene SCHEMBL18546560 0.95 HSD17B10 (0.75) HSD17B10ALDH1A1HPGDCYP1A2THRB
SCHEMBL2233815 0.95 HSD17B10 (0.75) HSD17B10ALDH1A1HPGDCYP1A2THRB
SCHEMBL4845945 0.95 HSD17B10 (0.75) HSD17B10ALDH1A1HPGDCYP1A2THRB
SCHEMBL4855087 0.92 HSD17B10 (0.71) HSD17B10ALDH1A1HPGDCYP1A2THRB
Chrysene SCHEMBL3747550 0.92 HPRT1 (0.78) HSD17B10ALDH1A1HPGDCYP1A2THRB
SCHEMBL4853390 0.92 HPRT1 (0.78) HSD17B10ALDH1A1HPGDCYP1A2THRB
SCHEMBL4846677 0.92 HPRT1 (0.78) HSD17B10ALDH1A1HPGDCYP1A2THRB
SCHEMBL4845629 0.92 HSD17B10 (0.89) HSD17B10ALDH1A1HPGDCYP1A2THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2582655-A1 LEAVING SUBSTITUENT-CONTAINING COMPOUND, ORGANIC SEMICONDUCTOR MATERIAL FORMED THEREFROM, ORGANIC ELECTRONIC DEVICE, ORGANIC THIN-FILM TRANSISTOR AND DISPLAY DEVICE USING THE ORGANIC SEMICONDUCTOR MATERIAL, METHOD FOR PRODUCING FILM-LIKE PRODUCT, PI-ELECTRON CONJUGATED COMPOUND AND METHOD FOR PRODUCING THE PI-ELECTRON CONJUGATED COMPOUND Ricoh Company, Ltd. (JP) 2013-04-24 EP disclosed
WO-2011158953-A1 LEAVING SUBSTITUENT-CONTAINING COMPOUND, ORGANIC SEMICONDUCTOR MATERIAL FORMED THEREFROM, ORGANIC ELECTRONIC DEVICE, ORGANIC THIN-FILM TRANSISTOR AND DISPLAY DEVICE USING THE ORGANIC SEMICONDUCTOR MATERIAL, METHOD FOR PRODUCING FILM-LIKE PRODUCT, PI-ELECTRON CONJUGATED COMPOUND AND METHOD FOR PRODUCING THE PI-ELECTRON CONJUGATED COMPOUND RICOH COMPANY, LTD. (JP) 2011-12-22 WO disclosed