SCHEMBL9998586

SCHEMBL9998586

O=C(OCc1ccccc1)c1cccc(CN2CN(c3ccccc3)C3(CCN(CCCn4c(C(=O)O)cc5ccccc54)CC3)C2=O)c1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.52
CYP3A4 P08684 2/20 0.52
CYP2D6 P10635 2/20 0.52
KMT2A Q03164 2/20 0.52
TP53 P04637 1/20 0.52
CYP1A2 P05177 1/20 0.52
MAPT P10636 1/20 0.52
ALOX15 P16050 1/20 0.52
TSHR P16473 1/20 0.52
MAPK1 P28482 1/20 0.52
CYP2C19 P33261 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
CYP2C9 P11712 1/20 0.44
F2 P00734 1/20 0.41
F10 P00742 1/20 0.41
OPRL1 P41146 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL318995 0.92 MEN1 (0.48) MEN1CYP3A4CYP2D6KMT2ATP53
SCHEMBL318868 0.86 MEN1 (0.52) MEN1CYP3A4CYP2D6KMT2ATP53
SCHEMBL318403 0.86 MEN1 (0.51) MEN1CYP3A4CYP2D6KMT2ATP53
SCHEMBL18601848 0.80 MEN1 (0.52) MEN1CYP3A4CYP2D6KMT2ATP53
SCHEMBL318729 0.79 MEN1 (0.54) MEN1CYP3A4CYP2D6KMT2ATP53
SCHEMBL318643 0.79 MEN1 (0.57) MEN1CYP3A4CYP2D6KMT2ATP53
SCHEMBL18601847 0.79 MEN1 (0.51) MEN1CYP3A4CYP2D6KMT2ATP53
SCHEMBL318623 0.79 MEN1 (0.51) MEN1CYP3A4CYP2D6KMT2ATP53
SCHEMBL319154 0.78 MEN1 (0.56) MEN1CYP3A4CYP2D6KMT2ATP53
SCHEMBL318732 0.78 MEN1 (0.53) MEN1CYP3A4CYP2D6KMT2ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2582701-A1 D2 ANTAGONISTS, METHODS OF SYNTHESIS AND METHODS OF USE Altos Therapeutics, LLC (US) 2013-04-24 EP disclosed
WO-2011160084-A1 D2 ANTAGONISTS, METHODS OF SYNTHESIS AND METHODS OF USE Altos Therapeutics, LLC (US) 2011-12-22 WO disclosed