SCHEMBL10016892

SCHEMBL10016892

CCc1ccc2cc(-c3c4ccccc4c(-c4ccc(-c5cncc(-c6ccccc6)c5)c5ccccc45)c4ccccc34)ccc2c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 11/20 0.45
CYP11B2 P19099 11/20 0.45
MAPT P10636 1/20 0.41
CYP1A2 P05177 2/20 0.40
CYP2A6 P11509 1/20 0.40
CYP19A1 P11511 2/20 0.36
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2B6 P20813 1/20 0.35
CYP2C19 P33261 1/20 0.35
GBA1 P04062 1/20 0.35
USP1 O94782 1/20 0.35
WDR48 Q8TAF3 1/20 0.35
MKNK1 Q9BUB5 1/20 0.34
MKNK2 Q9HBH9 1/20 0.34
MAPKAPK2 P49137 1/20 0.34
CYP17A1 P05093 1/20 0.33
PDE7A Q13946 1/20 0.33
PDE7B Q9NP56 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10016782 0.87 MAPT (0.48) CYP11B1CYP11B2MAPTCYP1A2CYP2A6
SCHEMBL10017119 0.87 MAPT (0.49) CYP11B1CYP11B2MAPTCYP1A2CYP2A6
SCHEMBL10016786 0.84 CYP1A2 (0.43) CYP11B1CYP11B2MAPTCYP1A2CYP2A6
SCHEMBL10017121 0.83 CYP1A2 (0.44) CYP11B1CYP11B2MAPTCYP1A2CYP2A6
SCHEMBL10016938 0.83 MAPT (0.36) CYP11B1CYP11B2MAPTCYP1A2CYP2A6
SCHEMBL10016886 0.82 MAPT (0.42) CYP11B1CYP11B2MAPTCYP1A2CYP2A6
SCHEMBL10017236 0.81 CYP1A2 (0.42) CYP11B1CYP11B2MAPTCYP1A2CYP2A6
SCHEMBL10016891 0.80 MAPKAPK2 (0.39) MAPTCYP1A2CYP2A6CYP3A4CYP2C9
SCHEMBL10016893 0.80 CYP1A2 (0.38) MAPTCYP1A2CYP2A6CYP3A4MAPKAPK2
SCHEMBL13015633 0.78 CYP11B1 (0.60) CYP11B1CYP11B2CYP1A2CYP19A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012005214-A1 ELECTRON TRANSPORT MATERIAL AND ORGANIC ELECTROLUMINESCENT ELEMENTS USING SAME JNC株式会社 (JP) 2012-01-12 WO disclosed