SCHEMBL10032047

SCHEMBL10032047

COc1ccc(-c2cc3nccc(C(C)C)c3s2)cn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K8 P41279 1/20 0.49
PIK3CA P42336 2/20 0.46
PIK3CG P48736 2/20 0.41
KCNH2 Q12809 1/20 0.41
PIK3CD O00329 1/20 0.41
PIP5K1C O60331 1/20 0.41
PIK3CB P42338 1/20 0.41
PI4KA P42356 1/20 0.41
PI4KB Q9UBF8 1/20 0.41
CDK4 P11802 1/20 0.40
CCND1 P24385 1/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
CYP2A6 P11509 2/20 0.40
KMT2A Q03164 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
CYP19A1 P11511 1/20 0.40
PDGFRB P09619 1/20 0.39
PDGFRA P16234 1/20 0.39
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15220094 0.84 MAP3K8 (0.53) MAP3K8PIK3CAPIK3CGKCNH2PIK3CD
SCHEMBL308582 0.82 MAP3K8 (0.51) MAP3K8PIK3CAPIK3CGKCNH2PIK3CD
SCHEMBL14953514 0.74 MAP3K8 (0.44) MAP3K8PIK3CAPIK3CGKCNH2PIK3CD
SCHEMBL7121628 0.73 NPC1 (0.47) MAP3K8PIK3CAKCNH2NPC1RAB9A
SCHEMBL13166726 0.71 MAP3K8 (0.42) MAP3K8PIK3CAPIK3CGPIK3CDPIP5K1C
SCHEMBL13975961 0.70 GRIN3B (0.46) CDK4CCND1GRIN3BGRIN1GRIN2C
SCHEMBL13976073 0.70 GRIN3B (0.46) CDK4CCND1GRIN3BGRIN1GRIN2C
SCHEMBL24837292 0.69 EGFR (0.39) PDGFRBPDGFRA
SCHEMBL24391687 0.69 KRAS (0.39)
SCHEMBL15220212 0.67 RAB9A (0.62) MAP3K8NPC1RAB9AKMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012008563-A1 NITROGENATED AROMATIC HETEROCYCLIC RING DERIVATIVE 協和発酵キリン株式会社 (JP) 2012-01-19 WO disclosed