SCHEMBL10042954

SCHEMBL10042954

COc1ccc(C2c3ccc(O)cc3OCC2c2ccc(C)cc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 5/20 0.55
ESR2 Q92731 5/20 0.55
EDNRB P24530 1/20 0.47
EDNRA P25101 1/20 0.47
ALDH1A1 P00352 1/20 0.43
ALOX15 P16050 2/20 0.43
ALOX12 P18054 2/20 0.43
MAPT P10636 2/20 0.43
MEN1 O00255 1/20 0.43
THRB P10828 1/20 0.43
KMT2A Q03164 1/20 0.43
MAPK1 P28482 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
ABCB1 P08183 2/20 0.40
MAOB P27338 2/20 0.40
LMNA P02545 2/20 0.40
CYP3A4 P08684 1/20 0.40
MAOA P21397 1/20 0.40
TP53 P04637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20831831 0.94 ESR1 (0.58) ESR1ESR2EDNRBEDNRAALDH1A1
SCHEMBL30362855 0.94 ESR1 (0.58) ESR1ESR2EDNRBEDNRAALDH1A1
SCHEMBL2604720 0.94 ESR1 (0.58) ESR1ESR2EDNRBEDNRAALDH1A1
SCHEMBL15312307 0.94 ESR1 (0.58) ESR1ESR2EDNRBEDNRAALDH1A1
SCHEMBL20831829 0.94 ESR1 (0.58) ESR1ESR2EDNRBEDNRAALDH1A1
SCHEMBL15013033 0.94 ESR1 (0.58) ESR1ESR2EDNRBEDNRAALDH1A1
SCHEMBL239999 0.94 ESR1 (0.58) ESR1ESR2EDNRBEDNRAALDH1A1
SCHEMBL19771459 0.93 ESR1 (0.50) ESR1ESR2EDNRBEDNRAALDH1A1
SCHEMBL24103714 0.91 ESR2 (0.52) ESR1ESR2ALDH1A1MAPTMEN1
SCHEMBL15006416 0.91 ESR2 (0.52) ESR1ESR2ALDH1A1MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120114766-A1 SUBSTITUTED CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY MARSHALL EDWARDS, INC. (US) 2012-05-10 US disclosed
US-20100130598-A1 METHODS FOR INDUCING PROGRAMMED CELL DEATH NOVOGEN RESEARCH PTY LTD. (AU) 2010-05-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120114766-A1 SUBSTITUTED CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY CDYL, XPA, TP53 ESR1 1328/4885ESR2 1134/4885EDNRB 4265/4885
US-20100130598-A1 METHODS FOR INDUCING PROGRAMMED CELL DEATH CASP3, BAX, BAD ESR1 4604/4885ESR2 3077/4885EDNRB 4059/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.