SCHEMBL10044440

SCHEMBL10044440

COc1cc(C)c(OCCN2CCOCC2)c(OC)c1

nearest known ligand 0.71

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SYK P43405 1/20 0.71
NPC1 O15118 1/20 0.54
TSHR P16473 2/20 0.53
CYP2D6 P10635 2/20 0.53
POLB P06746 1/20 0.53
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
ALDH1A1 P00352 3/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
BRD4 O60885 1/20 0.46
IL17A Q16552 1/20 0.46
PTPN1 P18031 1/20 0.45
CYP3A4 P08684 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15180060 0.84 SYK (0.63) SYKNPC1TSHRCYP2D6POLB
SCHEMBL10196165 0.83 SYK (1.00) SYKNPC1TSHRCYP2D6POLB
SCHEMBL12311750 0.80 NPC1 (0.70) SYKNPC1TSHRPOLBMEN1
SCHEMBL1911850 0.80 NPC1 (0.66) SYKNPC1TSHRPOLBMEN1
SCHEMBL12435658 0.80 SYK (0.77) SYKNPC1TSHRCYP2D6POLB
SCHEMBL348270 0.79 SYK (0.51) SYKNPC1TSHRCYP2D6POLB
SCHEMBL19227456 0.79 POLB (0.71) SYKNPC1CYP2D6POLBMEN1
SCHEMBL13791083 0.78 SYK (0.59) SYKNPC1TSHRALDH1A1SMN1; SMN2
SCHEMBL616988 0.78 BRD4 (0.51) SYKBRD4IL17A
SCHEMBL18639409 0.78 MAPK1 (0.47) ALDH1A1SMN1; SMN2BRD4PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012052420-A1 METHOD FOR PREPARING SUBSTITUTED N-(3-AMINO-QUINOXALIN-2-YL)-SULFONAMIDES AND THEIR INTERMEDIATES N-(3-CHLORO-QUINOXALIN-2-YL)SULFONAMIDES MERCK SERONO S.A. GENEVA (CH) 2012-04-26 WO disclosed