SCHEMBL10047889

SCHEMBL10047889

COC(=O)CCNC(=O)/C(C(=O)NCc1ccc(Cl)cc1)=C(/N)O

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.52
CYP2C19 P33261 2/20 0.49
CYP2C9 P11712 1/20 0.49
PLAAT3 P53816 2/20 0.46
PLAAT5 Q96KN8 2/20 0.46
PLAAT2 Q9NWW9 2/20 0.46
PLAAT4 Q9UL19 2/20 0.46
MAPT P10636 1/20 0.44
KMT2A Q03164 4/20 0.44
MEN1 O00255 3/20 0.44
TP53 P04637 1/20 0.43
HPGD P15428 1/20 0.43
GAA P10253 1/20 0.41
POLB P06746 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
LMNA P02545 1/20 0.41
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10047763 0.87 CYP2C19 (0.54) ALDH1A1CYP2C19CYP2C9PLAAT3PLAAT5
SCHEMBL15038458 0.80 ALDH1A1 (0.45) ALDH1A1CYP2C19CYP2C9PLAAT3PLAAT5
SCHEMBL10047770 0.77 CYP2C9 (0.51) ALDH1A1CYP2C19CYP2C9PLAAT3PLAAT5
SCHEMBL3635719 0.75 ALDH1A1 (0.51) ALDH1A1CYP2C19CYP2C9MAPTKMT2A
SCHEMBL15038479 0.74 CYP2C19 (0.44) ALDH1A1CYP2C19CYP2C9MAPTKMT2A
SCHEMBL15038438 0.72 CYP2C19 (0.40) ALDH1A1CYP2C19CYP2C9PLAAT3PLAAT5
SCHEMBL11068784 0.72 MEN1 (0.61) ALDH1A1CYP2C19CYP2C9PLAAT3PLAAT5
SCHEMBL17231391 0.71 CYP2C9 (0.72) ALDH1A1CYP2C19CYP2C9PLAAT3PLAAT5
SCHEMBL26764681 0.71 MEN1 (0.61) ALDH1A1CYP2C19CYP2C9MAPTKMT2A
SCHEMBL10055429 0.71 CYP2C9 (0.50) ALDH1A1CYP2C19CYP2C9MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020742-A1 NOVEL HETEROCYCLIC DERIVATIVES AND PHARMACEUTICAL COMPOSITION CONTAINING SAME 塩野義製薬株式会社 (JP) 2012-02-16 WO disclosed