SCHEMBL10050790

SCHEMBL10050790

CN1C(=O)c2c(c3c4cc(O[Si](C)(C)C(C)(C)C)ccc4[nH]c3c3ncc(F)cc23)C1=O

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 1/20 0.36
CHEK1 O14757 1/20 0.35
CA12 O43570 2/20 0.34
CA1 P00915 2/20 0.34
CA9 Q16790 2/20 0.34
GABRA1 P14867 1/20 0.34
GABRG2 P18507 1/20 0.34
GABRB3 P28472 1/20 0.34
KDM4E B2RXH2 4/20 0.33
ROCK2 O75116 2/20 0.33
JAK2 O60674 2/20 0.33
CDK4 P11802 2/20 0.33
CCND1 P24385 2/20 0.33
HSD17B10 Q99714 2/20 0.33
NPC1 O15118 1/20 0.32
ALDH1A1 P00352 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13609800 0.87 CDK4 (0.42) PDGFRBCHEK1CA12CA1CA9
SCHEMBL10075906 0.80 CHEK1 (0.52) CHEK1ROCK2
SCHEMBL10050791 0.71 CA12 (0.31) CA12CA1CA9
SCHEMBL8128221 0.69 PDGFRB (0.70) PDGFRBCHEK1KDM4EROCK2CDK4
SCHEMBL8113701 0.67 PDGFRB (0.49) PDGFRBCHEK1GABRA1GABRG2GABRB3
SCHEMBL5223967 0.66 MAOA (0.53) CA12CA1CA9KDM4EHSD17B10
SCHEMBL16504230 0.65 CDK4 (0.60) CHEK1GABRA1GABRG2GABRB3ROCK2
SCHEMBL23915925 0.64 MAOB (0.50) CA12CA1CA9
SCHEMBL28536275 0.62 CA12 (0.44) CA12CA1CA9KDM4EHSD17B10
SCHEMBL8125099 0.61 PDGFRB (0.54) PDGFRBKDM4EROCK2CDK4CCND1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8106039-B2 Metal complex phosphatidyl-inositol-3-kinase inhibitors THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2012-01-31 US disclosed