Rocaglamide

Rocaglamide

SCHEMBL10054686

COc1ccc([C@]23Oc4cc(OC)cc(OC)c4[C@]2(O)[C@H](O)[C@H](C(=O)N(C)C)[C@@H]3c2ccccc2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EIF4A1 P60842 18/20 1.00
NFKB1 P19838 1/20 1.00
RELA Q04206 1/20 1.00
CYP3A4 P08684 1/20 0.80
HIF1A Q16665 1/20 0.80
PAX8 Q06710 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Rocaglamide SCHEMBL29439568 1.00 EIF4A1 (1.00) EIF4A1NFKB1RELACYP3A4HIF1A
Rocaglamide SCHEMBL751061 1.00 EIF4A1 (1.00) EIF4A1NFKB1RELACYP3A4HIF1A
Rocaglamide SCHEMBL752144 1.00 EIF4A1 (1.00) EIF4A1NFKB1RELACYP3A4HIF1A
Rocaglamide SCHEMBL20386162 1.00 EIF4A1 (1.00) EIF4A1NFKB1RELACYP3A4HIF1A
Rocaglamide SCHEMBL29407815 1.00 EIF4A1 (1.00) EIF4A1NFKB1RELACYP3A4HIF1A
Rocaglamide SCHEMBL24127774 1.00 EIF4A1 (1.00) EIF4A1NFKB1RELACYP3A4HIF1A
SCHEMBL12182311 0.93 EIF4A1 (0.87) EIF4A1NFKB1RELACYP3A4HIF1A
SCHEMBL29370550 0.91 EIF4A1 (0.84) EIF4A1NFKB1RELACYP3A4HIF1A
SCHEMBL15079078 0.91 EIF4A1 (0.86) EIF4A1NFKB1RELACYP3A4HIF1A
Rocagloic Acid SCHEMBL750035 0.91 EIF4A1 (0.86) EIF4A1NFKB1RELACYP3A4HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037062-A2 NEW ROUTE TO SYNTHETIC ANALOGUES OF ROCAGLAMIDE AND AGLAFOLINE USING CASCADE TRANSFORMATIONS INITIATED BY OXY-COPE REARRANGEMENTS OF BIS-ALKYNES FLORIDA STATE UNIVERSITY RESEARCH FOUNDATION, INC. (US) 2012-03-22 WO disclosed