SCHEMBL10057488

SCHEMBL10057488

Cc1ccc(-c2ccc(-c3ccc(-c4nc(-c5ccc(-c6ccccc6)cc5)nc(-c5ccc(-c6ccccc6)cc5)n4)cc3)cc2)nc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.53
CYP2A6 P11509 1/20 0.53
L3MBTL1 Q9Y468 2/20 0.50
CCR1 P32246 1/20 0.50
CCR5 P51681 1/20 0.50
CCR8 P51685 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
MEN1 O00255 5/20 0.47
KMT2A Q03164 5/20 0.47
ALDH1A1 P00352 3/20 0.47
MAPT P10636 2/20 0.47
HPGD P15428 2/20 0.47
LDHA P00338 1/20 0.46
KDM4E B2RXH2 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
NPC1 O15118 4/20 0.44
RAB9A P51151 4/20 0.44
SLC2A1 P11166 1/20 0.44
ALDH1A3 P47895 1/20 0.44
BAZ2B Q9UIF8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17532913 0.94 MEN1 (0.48) CYP3A4CYP2A6L3MBTL1CCR1CCR5
SCHEMBL18325218 0.92 L3MBTL1 (0.48) CYP3A4CYP2A6L3MBTL1MEN1KMT2A
SCHEMBL12359222 0.91 CYP3A4 (0.61) CYP3A4CYP2A6L3MBTL1CCR1CCR5
SCHEMBL11976414 0.90 L3MBTL1 (0.50) CYP3A4CYP2A6L3MBTL1MEN1KMT2A
SCHEMBL12628224 0.89 CCR1 (0.54) CYP3A4CYP2A6L3MBTL1CCR1CCR5
SCHEMBL21729301 0.89 CYP3A4 (0.47) CYP3A4CYP2A6L3MBTL1CCR1CCR5
SCHEMBL404433 0.87 CYP3A4 (0.66) CYP3A4CYP2A6L3MBTL1CCR1CCR5
SCHEMBL18267900 0.87 CYP3A4 (0.50) CYP3A4CYP2A6L3MBTL1CCR1CCR5
SCHEMBL18325353 0.86 MEN1 (0.50) CYP3A4L3MBTL1MEN1KMT2AALDH1A1
SCHEMBL21202993 0.86 MEN1 (0.50) CYP3A4L3MBTL1MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130264561-A1 ELECTROACTIVE COMPOSITIONS FOR ELECTRONIC APPLICATIONS E I DU PONT DE NEMOURS AND COMPANY (US) 2013-10-10 US disclosed
US-20130264561-A1 ELECTROACTIVE COMPOSITIONS FOR ELECTRONIC APPLICATIONS E I DU PONT DE NEMOURS AND COMPANY (US) 2013-10-10 US disclosed
US-20130264560-A1 TRIAZINE DERIVATIVES FOR ELECTRONIC APPLICATIONS E I DU PONT DE NEMOURS AND COMPANY (US) 2013-10-10 US disclosed
US-20130264560-A1 TRIAZINE DERIVATIVES FOR ELECTRONIC APPLICATIONS E I DU PONT DE NEMOURS AND COMPANY (US) 2013-10-10 US disclosed
WO-2012087961-A2 ELECTROACTIVE COMPOSITIONS FOR ELECTRONIC APPLICATIONS E. I. DU PONT DE NEMOURS AND COMPANY (US) 2012-06-28 WO disclosed
WO-2012087960-A1 TRIAZINE DERIVATIVES FOR ELECTRONIC APPLICATIONS E. I. DU PONT DE NEMOURS AND COMPANY (US) 2012-06-28 WO disclosed