SCHEMBL10065029

SCHEMBL10065029

CN(C)C1(Cc2ccccc2)CCC2(CC1)c1[nH]c3ccccc3c1CCN2C(=O)c1c(N)cccc1Cl

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 7/20 0.50
OGFRL1 Q5TC84 3/20 0.50
OPRL1 P41146 3/20 0.43
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
F12 P00748 2/20 0.34
TRPV1 Q8NER1 2/20 0.34
TRPA1 O75762 2/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
OPRD1 P41143 2/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
OPRK1 P41145 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2141647 0.94 OPRM1 (0.54) OPRM1OGFRL1OPRL1KMT2AMEN1
SCHEMBL2141136 0.86 OPRM1 (0.54) OPRM1OGFRL1OPRL1KMT2AMEN1
SCHEMBL2140032 0.85 OPRM1 (0.54) OPRM1OGFRL1OPRL1KMT2AMEN1
SCHEMBL2141981 0.82 OPRM1 (0.49) OPRM1OGFRL1OPRL1KMT2ATRPV1
SCHEMBL2139574 0.82 OPRM1 (0.54) OPRM1OGFRL1OPRL1KMT2AMEN1
SCHEMBL2140335 0.81 OPRM1 (0.58) OPRM1OGFRL1OPRL1KMT2AMEN1
SCHEMBL2141092 0.81 OPRM1 (0.52) OPRM1OGFRL1OPRL1KMT2ATRPV1
SCHEMBL2142688 0.80 OPRM1 (0.54) OPRM1OGFRL1OPRL1KMT2AMEN1
SCHEMBL2142957 0.80 OPRM1 (0.52) OPRM1OGFRL1OPRL1KMT2AMEN1
SCHEMBL2137582 0.80 OPRM1 (0.52) OPRM1OGFRL1OPRL1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1868600-B1 SPIROCYCLIC CYCLOHEXANE DERIVATIVES FOR USE IN THE TREATMENT OF SUBSTANCE DEPENDENCY GRUENENTHAL GMBH (DE) 2012-06-27 EP disclosed