SCHEMBL10068458

SCHEMBL10068458

CC(=O)C(N)Cc1c[nH]c2c(C)cccc12

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SOS2 Q07890 1/20 0.68
HTR2A P28223 1/20 0.55
MAPT P10636 3/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
NPSR1 Q6W5P4 1/20 0.54
BRPF1 P55201 1/20 0.52
NR3C1 P04150 2/20 0.48
KDM4E B2RXH2 1/20 0.48
MEN1 O00255 1/20 0.48
LMNA P02545 1/20 0.48
MPO P05164 1/20 0.48
TSHR P16473 1/20 0.48
BLM P54132 1/20 0.48
PMP22 Q01453 1/20 0.48
KMT2A Q03164 1/20 0.48
HIF1A Q16665 1/20 0.48
NR4A2 P43354 1/20 0.46
PGR P06401 1/20 0.46
NR3C2 P08235 1/20 0.46
TNF P01375 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29405720 0.89 SOS2 (0.68) SOS2HTR2AMAPTSMN1; SMN2NPSR1
SCHEMBL2033276 0.89 SOS2 (0.68) SOS2HTR2AMAPTSMN1; SMN2NPSR1
SCHEMBL10023253 0.89 SOS2 (0.68) SOS2HTR2AMAPTSMN1; SMN2NPSR1
SCHEMBL31369774 0.89 SOS2 (0.68) SOS2HTR2AMAPTSMN1; SMN2NPSR1
SCHEMBL2033277 0.89 SOS2 (0.68) SOS2HTR2AMAPTSMN1; SMN2NPSR1
SCHEMBL23859779 0.85 SOS2 (0.63) SOS2HTR2AMAPTSMN1; SMN2NPSR1
SCHEMBL10849704 0.85 SOS2 (0.63) SOS2HTR2AMAPTSMN1; SMN2NPSR1
SCHEMBL19846987 0.85 SOS2 (0.48) SOS2HTR2AMAPTSMN1; SMN2NPSR1
SCHEMBL19846988 0.85 HTR2A (0.54) SOS2HTR2AMAPTSMN1; SMN2KDM4E
SCHEMBL24042700 0.81 SOS2 (0.57) SOS2HTR2AMAPTSMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012173846-A2 PEPTIDOMIMETIC MACROCYCLES AILERON THERAPEUTICS, INC. (US) 2012-12-20 WO disclosed
WO-2012021876-A2 PEPTIDOMIMETIC MACROCYCLES AILERON THERAPEUTICS, INC. (US) 2012-02-16 WO disclosed
WO-2012021875-A1 PEPTIDOMIMETIC MACROCYCLES WITH TRIAZOLE LINKERS AILERON THERAPEUTICS, INC. (US) 2012-02-16 WO disclosed