SCHEMBL10073787

SCHEMBL10073787

O=C(Nc1ccccc1)Nc1ccc(Oc2ncnc3cc(F)ccc23)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 11/20 1.00
KDR P35968 7/20 0.69
RAF1 P04049 1/20 0.65
PDGFRB P09619 1/20 0.65
KIT P10721 1/20 0.65
FLT1 P17948 1/20 0.65
FLT4 P35916 1/20 0.65
BRAF P15056 2/20 0.64
MAPK14 Q16539 1/20 0.64
TNNI3K Q59H18 1/20 0.64
POLB P06746 1/20 0.62
SAE1 Q9UBE0 1/20 0.62
UBA2 Q9UBT2 1/20 0.62
FLT3 P36888 2/20 0.61
AURKB Q96GD4 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22548175 0.87 CSF1R (1.00) CSF1RKDRRAF1PDGFRBKIT
SCHEMBL22548458 0.87 CSF1R (0.78) CSF1RKDRRAF1PDGFRBKIT
SCHEMBL717412 0.87 CSF1R (0.77) CSF1RKDRPOLBSAE1UBA2
SCHEMBL22533942 0.84 CSF1R (1.00) CSF1RAURKB
SCHEMBL31236177 0.84 CSF1R (1.00) CSF1RAURKB
SCHEMBL10073792 0.84 CSF1R (0.73) CSF1RKDRRAF1PDGFRBKIT
SCHEMBL282549 0.84 CSF1R (0.72) CSF1RKDRRAF1PDGFRBKIT
SCHEMBL22548194 0.84 CSF1R (0.82) CSF1RKDRAURKB
SCHEMBL22548172 0.84 CSF1R (0.83) CSF1RAURKB
SCHEMBL22548453 0.83 CSF1R (1.00) CSF1RKDRRAF1PDGFRBKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220213064-A1 HETEROCYCLIC COMPOUNDS AS KINASE INHIBITORS FOR THERAPEUTIC USES NATIONAL HEALTH RESEARCH INSTITUTES (TW) 2022-07-07 US disclosed
WO-2020210481-A1 HETEROCYCLIC COMPOUNDS AS KINASE INHIBITORS FOR THERAPEUTIC USES NATION HEALTH RESEARCH INSTITUTES (TW) 2020-10-15 WO disclosed
US-8957087-B2 Heterocyclic substituted acardite derivate and application thereof Jiangsu Provincial Institute of Materia Medica Co., Ltd. (CN) 2015-02-17 US disclosed
US-20120053192-A1 Heterocyclic Substituted Acardite Derivate and Application Thereof NANJING LUYESIKE PHARMACEUTICAL CO., LTD. (CN) 2012-03-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120053192-A1 Heterocyclic Substituted Acardite Derivate and Application Thereof H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, IDH1, CA7 CSF1R 2180/4885KDR 3633/4885RAF1 955/4885
US-20220213064-A1 HETEROCYCLIC COMPOUNDS AS KINASE INHIBITORS FOR THERAPEUTIC USES MCL1, KIT, CHUK CSF1R 6/4885KDR 80/4885RAF1 15/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.