SCHEMBL10073792

SCHEMBL10073792

Cc1cc2c(Oc3ccc(NC(=O)Nc4ccccc4)cc3)ncnc2cc1F

nearest known ligand 0.73

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 8/20 0.73
KDR P35968 12/20 0.70
PDGFRA P16234 2/20 0.61
BRAF P15056 2/20 0.59
KIT P10721 3/20 0.58
RAF1 P04049 2/20 0.58
PDGFRB P09619 2/20 0.58
FLT1 P17948 2/20 0.58
FLT4 P35916 2/20 0.58
MET P08581 1/20 0.58
SRC P12931 1/20 0.58
MAPK14 Q16539 1/20 0.58
TNNI3K Q59H18 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL282170 0.85 KDR (0.62) CSF1RKDRPDGFRABRAFRAF1
SCHEMBL10073787 0.84 CSF1R (1.00) CSF1RKDRBRAFKITRAF1
SCHEMBL281945 0.84 KDR (0.57) CSF1RKDRPDGFRABRAFKIT
SCHEMBL22548175 0.81 CSF1R (1.00) CSF1RKDRPDGFRABRAFKIT
SCHEMBL22548458 0.79 CSF1R (0.78) CSF1RKDRBRAFKITRAF1
SCHEMBL7479842 0.79 KDR (0.81) CSF1RKDRPDGFRABRAFKIT
SCHEMBL22533942 0.79 CSF1R (1.00) CSF1R
SCHEMBL31236177 0.79 CSF1R (1.00) CSF1R
SCHEMBL5202625 0.78 KDR (0.81) CSF1RKDRPDGFRABRAFKIT
SCHEMBL5202980 0.77 KDR (0.85) CSF1RKDRPDGFRABRAFKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8957087-B2 Heterocyclic substituted acardite derivate and application thereof Jiangsu Provincial Institute of Materia Medica Co., Ltd. (CN) 2015-02-17 US disclosed
US-20120053192-A1 Heterocyclic Substituted Acardite Derivate and Application Thereof NANJING LUYESIKE PHARMACEUTICAL CO., LTD. (CN) 2012-03-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120053192-A1 Heterocyclic Substituted Acardite Derivate and Application Thereof H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, IDH1, CA7 CSF1R 2180/4885KDR 3633/4885PDGFRA 1115/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.