SCHEMBL10074897

SCHEMBL10074897

Cc1ccc(-c2nnn(C)c2/C=C/c2nc(C)c(C(=O)NC3CCOCC3)s2)cc1

nearest known ligand 0.87

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 12/20 0.87
ITGA5 P08648 1/20 0.41
CNR1 P21554 2/20 0.39
ALDH1A1 P00352 2/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
CHRM4 P08173 1/20 0.37
TSHR P16473 1/20 0.36
PPARG P37231 1/20 0.36
PPARD Q03181 1/20 0.36
PPARA Q07869 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4407571 0.93 GABRA5 (1.00) GABRA5ALDH1A1LMNAHTTCHRM4
SCHEMBL4410068 0.85 GABRA5 (1.00) GABRA5ITGA5ALDH1A1LMNAHTT
SCHEMBL4402982 0.76 GABRA5 (1.00) GABRA5CHRM4PPARDPPARA
SCHEMBL2683793 0.75 GABRA5 (1.00) GABRA5CNR1ALDH1A1NPC1RAB9A
SCHEMBL2683802 0.75 GABRA5 (1.00) GABRA5CNR1ALDH1A1NPC1RAB9A
SCHEMBL2683796 0.74 GABRA5 (0.75) GABRA5ALDH1A1LMNATSHRPPARA
SCHEMBL2685284 0.73 GABRA5 (0.77) GABRA5ALDH1A1NPC1RAB9A
SCHEMBL2685279 0.73 GABRA5 (0.77) GABRA5ALDH1A1NPC1RAB9A
SCHEMBL16290095 0.72 GABRA5 (0.76) GABRA5ITGA5ALDH1A1RAB9A
SCHEMBL2689993 0.71 GABRA5 (0.65) GABRA5ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012062623-A1 TRIAZOLE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS F. HOFFMANN-LA ROCHE AG (CH) 2012-05-18 WO disclosed