SCHEMBL10075909

SCHEMBL10075909

BC1=C(c2c(-c3ccc(F)cn3)[nH]c3ccc(O)cc23)C(=O)N(C)C1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 4/20 0.37
WEE1 P30291 2/20 0.37
TGFBR1 P36897 1/20 0.36
TGFBR2 P37173 1/20 0.36
MEN1 O00255 1/20 0.34
POLB P06746 1/20 0.34
GAA P10253 1/20 0.34
CASP6 P55212 1/20 0.34
KMT2A Q03164 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
PRKD1 Q15139 1/20 0.34
CDK5 Q00535 2/20 0.34
CDK5R1 Q15078 2/20 0.34
NR1I2 O75469 1/20 0.33
MAPT P10636 1/20 0.33
GABRP O00591 1/20 0.33
GABRD O14764 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRB1 P18505 1/20 0.33
GABRG2 P18507 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10050791 0.71 CA12 (0.31) TGFBR1TGFBR2GSK3B
SCHEMBL10075906 0.66 CHEK1 (0.52) CHEK1WEE1CDK5CDK5R1GSK3B
SCHEMBL10075907 0.62 CDK5 (0.55) CDK5CDK5R1MAPTFLT3CYP1A1
SCHEMBL27549068 0.61 NR1I2 (0.68) CHEK1WEE1MEN1POLBGAA
SCHEMBL20685664 0.59 ACHE (0.55) CHEK1WEE1MEN1POLBGAA
SCHEMBL12987394 0.59 NPC1 (0.53) MEN1POLBKMT2AMAPTALK
SCHEMBL6506227 0.58 WEE1 (0.48) CHEK1WEE1MEN1POLBGAA
SCHEMBL12987550 0.57 ESR1 (0.46) FEN1
SCHEMBL15797297 0.56 GSK3B (0.64) MEN1GAAKMT2AMAPTGSK3B
SCHEMBL27048226 0.56 CHEK1 (0.56) CHEK1WEE1CDK5CDK5R1GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8106039-B2 Metal complex phosphatidyl-inositol-3-kinase inhibitors THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2012-01-31 US disclosed