SCHEMBL10077002

SCHEMBL10077002

CCOC(=O)c1ccc(NC(=O)CC2Nc3cccc4cccc(c34)NC2=O)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 16/20 1.00
GAA P10253 12/20 1.00
TP53 P04637 4/20 1.00
THRB P10828 1/20 1.00
MEN1 O00255 8/20 0.76
KMT2A Q03164 8/20 0.76
ALDH1A1 P00352 7/20 0.76
POLB P06746 4/20 0.76
KDM4E B2RXH2 4/20 0.76
BLM P54132 3/20 0.76
PLEC Q15149 2/20 0.76
MAPK1 P28482 1/20 0.76
MCL1 Q07820 1/20 0.76
L3MBTL1 Q9Y468 1/20 0.76
CYP1A2 P05177 2/20 0.73
CYP3A4 P08684 2/20 0.73
CYP2C9 P11712 2/20 0.73
CYP2C19 P33261 2/20 0.73
GFER P55789 1/20 0.73
LMNA P02545 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10077846 0.87 MAPT (1.00) MAPTGAATP53THRBMEN1
SCHEMBL10077924 0.86 MAPT (1.00) MAPTGAATP53THRBMEN1
SCHEMBL10077404 0.85 MAPT (1.00) MAPTGAATP53THRBMEN1
SCHEMBL10077845 0.82 GAA (1.00) MAPTGAATP53THRBMEN1
SCHEMBL10077844 0.81 MAPT (1.00) MAPTGAATP53THRBMEN1
SCHEMBL13166883 0.69 MST1R (1.00) MAPTGAATP53MEN1KMT2A
SCHEMBL6689489 0.68 TSHR (0.72) MAPTGAATP53MEN1KMT2A
SCHEMBL5807379 0.68 TSHR (0.72) MAPTGAATP53MEN1KMT2A
SCHEMBL9671985 0.68 TSHR (0.77) MAPTGAATP53MEN1KMT2A
SCHEMBL7494835 0.67 MAPT (0.63) MAPTGAATP53MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012016133-A2 ROS1 KINASE INHIBITORS FOR THE TREATMENT OF GLIOBLASTOMA AND OTHER P53-DEFICIENT CANCERS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2012-02-02 WO disclosed